SCHEMBL6507408

SCHEMBL6507408

O=C1CN(C(=O)OCc2ccccc2)C(=O)CN1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.61
RAB9A P51151 3/20 0.61
SMN1; SMN2 Q16637 3/20 0.61
GAA P10253 2/20 0.61
MAPK1 P28482 1/20 0.61
L3MBTL1 Q9Y468 1/20 0.49
HTR2C P28335 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
GLA P06280 1/20 0.43
CTRB1 P17538 1/20 0.43
P2RX4 Q99571 2/20 0.43
PARP1 P09874 1/20 0.42
DDB1 Q16531 1/20 0.42
CRBN Q96SW2 1/20 0.42
CYP2C19 P33261 1/20 0.42
P2RX1 P51575 1/20 0.42
P2RX3 P56373 1/20 0.42
ALDH1A1 P00352 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29235094 0.85 NPC1 (0.61) NPC1RAB9ASMN1; SMN2GAAMAPK1
SCHEMBL3490697 0.78 ALDH1A1 (0.45) NPC1RAB9ASMN1; SMN2GAAMAPK1
SCHEMBL3767544 0.78 NPC1 (0.52) NPC1RAB9ASMN1; SMN2GAAMAPK1
SCHEMBL8522162 0.77 SMN1; SMN2 (0.56) NPC1RAB9ASMN1; SMN2GAAMAPK1
SCHEMBL1570950 0.76 NPC1 (0.50) NPC1RAB9ASMN1; SMN2GAAMAPK1
SCHEMBL11860696 0.75 GAA (0.63) NPC1RAB9ASMN1; SMN2GAAMAPK1
SCHEMBL92518 0.75 L3MBTL1 (0.56) NPC1RAB9ASMN1; SMN2GAAMAPK1
SCHEMBL2539997 0.75 NPC1 (0.67) NPC1RAB9ASMN1; SMN2GAAMAPK1
SCHEMBL20122609 0.73 NPC1 (0.53) NPC1RAB9ASMN1; SMN2GAAMAPK1
SCHEMBL3074986 0.73 MEN1 (0.52) NPC1RAB9ASMN1; SMN2GAAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005082866-A2 SUBSTITUTED 1, 2, 4- TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS PFIZER LIMITED (GB) 2005-09-09 WO claimed
WO-2005082866-A2 SUBSTITUTED 1, 2, 4- TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS PFIZER LIMITED (GB) 2005-09-09 WO disclosed