SCHEMBL6507594

SCHEMBL6507594

Cc1sc(-c2ccccc2Cl)nc1C(=O)NCc1cc(CC(OC(C)C)C(=O)O)ccc1-c1ccco1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.38
ADORA1 P30542 4/20 0.38
ADORA3 P0DMS8 3/20 0.38
ADORA2B P29275 3/20 0.38
ALDH1A1 P00352 5/20 0.38
KDM4E B2RXH2 3/20 0.38
PPARG P37231 3/20 0.36
PPARD Q03181 3/20 0.36
PPARA Q07869 3/20 0.36
MAPT P10636 5/20 0.35
KMT2A Q03164 4/20 0.35
MEN1 O00255 3/20 0.35
HSD17B10 Q99714 2/20 0.35
POLB P06746 2/20 0.35
RECQL P46063 2/20 0.35
MCL1 Q07820 2/20 0.35
ALOX15 P16050 1/20 0.35
APEX1 P27695 1/20 0.35
BCL2L1 Q07817 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6505714 0.90 NPC1 (0.41) ADORA2AADORA1ADORA3ADORA2BALDH1A1
SCHEMBL6496502 0.86 PPARA (0.39) ALDH1A1PPARGPPARDPPARAMAPT
SCHEMBL6505578 0.84 PPARG (0.41) PPARGPPARDPPARA
SCHEMBL6503008 0.83 PPARG (0.48) PPARGPPARDPPARA
SCHEMBL6506146 0.81 EPHX2 (0.37) PPARGPPARDPPARA
Trifluoroacetic Acid SCHEMBL6505587 0.81 PPARA (0.38) ADORA2AADORA1ALDH1A1PPARGPPARD
SCHEMBL6495630 0.80 PPARA (0.38) ALDH1A1PPARGPPARDPPARAMAPT
SCHEMBL6496468 0.79 MAPT (0.38) ADORA2AADORA1ALDH1A1PPARGPPARD
SCHEMBL7684246 0.79 SHMT1 (0.39) KDM4EPPARGPPARDPPARAMAPT
SCHEMBL6496963 0.78 TP53 (0.39) ADORA2AADORA1ADORA3ADORA2BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed