SCHEMBL6508399

SCHEMBL6508399

Oc1cc(C2=C(c3ccc(F)cc3)[N]C(=S)N2)ccn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38
ATM Q13315 1/20 0.38
ALDH1A1 P00352 2/20 0.37
MAPT P10636 2/20 0.37
HPGD P15428 2/20 0.37
GFER P55789 1/20 0.37
GSK3B P49841 2/20 0.33
CCNB2 O95067 1/20 0.33
CDK1 P06493 1/20 0.33
CCNB1 P14635 1/20 0.33
GSK3A P49840 1/20 0.33
CDK5 Q00535 1/20 0.33
CDK5R1 Q15078 1/20 0.33
CCNB3 Q8WWL7 1/20 0.33
MAPK10 P53779 2/20 0.31
TGFBR1 P36897 1/20 0.31
MAPK14 Q16539 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2295783 0.86 MAPK14 (0.41) ALDH1A1MAPTHPGDGFERGSK3B
SCHEMBL2299116 0.80 MAPK14 (0.42) ALDH1A1MAPTHPGDGSK3BMAPK10
SCHEMBL2298729 0.73 MAPK14 (0.53) GSK3BMAPK14MAPK13MAPK12MAPK11
SCHEMBL4096702 0.71 MAPK14 (0.44) MEN1NPC1RAB9AKMT2AATM
SCHEMBL6515232 0.69 MAPK14 (0.41) MAPTGSK3BCCNB2CDK1CCNB1
SCHEMBL5253575 0.62 MAPK14 (0.45) MEN1NPC1RAB9AKMT2AATM
SCHEMBL608871 0.60
SCHEMBL28673160 0.60 CYP2A6 (0.49) MAPTGSK3AMAPK14ALKCYP3A4
SCHEMBL6408354 0.60 MAPK10 (0.55) MEN1NPC1RAB9AKMT2AATM
SCHEMBL27157236 0.59 NPC1 (0.56) MEN1NPC1RAB9AKMT2AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005105813-A1 IMPROVED PROCESS FOR THE MANUFACTURE OF CEFTRIAXONE SODIUM WOCKHARDT LIMITED (IN) 2005-11-10 WO claimed
WO-2005105814-A1 TETRACYCLIC INHIBITORS OF JANUS KINASES INCYTE CORPORATION (US) 2005-11-10 WO disclosed