SCHEMBL6508909

SCHEMBL6508909

CCCCCc1ccc(NC(N)=Nc2nc(C)c3c(n2)CCCC3)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.61
RAB9A P51151 1/20 0.61
SPHK1 Q9NYA1 7/20 0.41
MAPT P10636 2/20 0.41
CRHBP P24387 2/20 0.41
CRHR2 Q13324 2/20 0.41
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2A Q12879 1/20 0.41
GRIN2B Q13224 1/20 0.41
GRIN2C Q14957 1/20 0.41
GRIN3A Q8TCU5 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
NPC1 O15118 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
STAT3 P40763 1/20 0.41
RECQL P46063 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5923382 0.77 MEN1 (0.42) RAB9ASPHK1MAPTNPC1
SCHEMBL6510623 0.75 RAB9A (0.67) MAPK1RAB9ASPHK1CRHBPCRHR2
SCHEMBL4985481 0.74 GRIN2D (0.68) MAPK1RAB9ASPHK1GRIN2DGRIN3B
SCHEMBL6517381 0.71 SMN1; SMN2 (0.53) MAPK1RAB9AMAPTCRHBPCRHR2
SCHEMBL4980238 0.71 SIGMAR1 (0.71) MAPK1RAB9AGRIN2DGRIN3BGRIN1
SCHEMBL4113089 0.70 MAPT (0.46) MAPK1RAB9AMAPTCRHBPCRHR2
SCHEMBL5923235 0.66 KDM4E (0.39) RAB9AMAPTNPC1CYP1A2
SCHEMBL1955157 0.64 THRA (0.63) SPHK1
SCHEMBL3428500 0.64 THRA (0.55) RAB9ASPHK1NPC1
SCHEMBL4979877 0.64 SIGMAR1 (0.62) MAPK1RAB9AGRIN2DGRIN3BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005095345-A2 HETEROARYL GUANIDINES AS INHIBITORS OF VIRAL REPLICATION ACHILLION PHARMACEUTICALS, INC. (US) 2005-10-13 WO claimed