SCHEMBL6509129

SCHEMBL6509129

COC(=O)CCCn1c(=O)c2c(C)n[nH]c2c2cc(Br)cc(C3CCCCO3)c21

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
DYRK1A Q13627 2/20 0.32
CASP3 P42574 1/20 0.31
CHEK1 O14757 1/20 0.31
KCNH2 Q12809 1/20 0.31
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6513337 0.75 PIK3R1 (0.45) ALDH1A1DYRK1ACASP3CHEK1CNR2
SCHEMBL6525537 0.70 CASP3 (0.37) HPGDALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL6508143 0.65 PIK3R1 (0.43) ALDH1A1CHEK1CNR2
SCHEMBL6525512 0.60 MAPT (0.51) ALDH1A1CYP1A2CYP3A4CYP2C19CNR2
SCHEMBL6508464 0.60 CHEK1 (0.53) HPGDALDH1A1CHEK1KCNH2CNR2
SCHEMBL6507976 0.59 CHEK1 (0.53) ALDH1A1CHEK1KCNH2CNR2
SCHEMBL6522871 0.57 CHEK1 (0.51) ALDH1A1CHEK1KCNH2
SCHEMBL6519279 0.57 SYK (0.43)
SCHEMBL31072035 0.55 HPGD (0.43) HPGD
SCHEMBL21767502 0.55 HPGD (0.43) HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005028474-A2 PYRAZOLOQUINOLINE DERIVATIVES AS CHK-1 INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2005-03-31 WO disclosed