SCHEMBL6525537

SCHEMBL6525537

COC(=O)CCCn1c(=O)c2c(C)nn(C3CCCCO3)c2c2cc(Br)ccc21

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.37
CNR2 P34972 7/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C19 P33261 1/20 0.37
DYRK1A Q13627 3/20 0.36
CDK1 P06493 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
MAPK8 P45983 2/20 0.33
TLR4 O00206 1/20 0.33
RXRA P19793 1/20 0.33
RXRB P28702 1/20 0.33
RXRG P48443 1/20 0.33
CNR1 P21554 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6523707 0.75 TOP1 (0.41) CNR2
SCHEMBL6513337 0.73 PIK3R1 (0.45) CASP3CNR2ALDH1A1DYRK1ACDK1
SCHEMBL6508889 0.72 ATR (0.42) CNR2DYRK1A
SCHEMBL18281904 0.71 GAA (0.41) CNR2ALDH1A1HPGDCYP2C19MAPK8
SCHEMBL6523125 0.71 PTGS2 (0.38) ALDH1A1HPGDSMN1; SMN2
SCHEMBL6509129 0.70 HPGD (0.33) CASP3CNR2ALDH1A1HPGDCYP1A2
SCHEMBL6510884 0.69 CHEK1 (0.56) CASP3CNR2ALDH1A1DYRK1ACDK1
SCHEMBL6502931 0.69 ELANE (0.51) CNR2ALDH1A1HPGDCDK1MAPK8
SCHEMBL29593200 0.69 ELANE (0.51) CNR2ALDH1A1HPGDCDK1MAPK8
SCHEMBL23219108 0.69 RXRA (0.39) CNR2ALDH1A1CDK1MAPK8RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050245563-A1 Chk-1 inhibitors MILLENNIUM PHARMACEUTICALS, INC. (US) 2005-11-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050245563-A1 Chk-1 inhibitors CHKA, CHKB, CHEK1 CASP3 3036/4885CNR2 3139/4885ALDH1A1 4635/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.