SCHEMBL6511364

SCHEMBL6511364

COC(=O)[C@@H](CC(C)C)Nc1nc(Cl)cc(Sc2ccc(OC)cc2)n1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPR3 P17342 3/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
TAS1R3 Q7RTX0 7/20 0.42
TAS1R1 Q7RTX1 7/20 0.42
NOS3 P29474 2/20 0.38
NOS1 P29475 2/20 0.38
NOS2 P35228 2/20 0.38
ELANE P08246 5/20 0.37
MAPT P10636 1/20 0.37
ANPEP P15144 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6511358 1.00 NPR3 (0.45) NPR3CYP2C9CYP2C19TAS1R3TAS1R1
SCHEMBL8297653 0.84 TAS1R3 (0.43) NPR3CYP2C9CYP2C19TAS1R3TAS1R1
SCHEMBL6512169 0.82 NPR3 (0.47) NPR3CYP2C9CYP2C19TAS1R3TAS1R1
SCHEMBL6512165 0.82 NPR3 (0.47) NPR3CYP2C9CYP2C19TAS1R3TAS1R1
SCHEMBL6508225 0.81 NPR3 (0.60) NPR3CYP2C9CYP2C19TAS1R3TAS1R1
SCHEMBL6508232 0.81 NPR3 (0.60) NPR3CYP2C9CYP2C19TAS1R3TAS1R1
SCHEMBL6507666 0.80 HPGD (0.48) MAPT
SCHEMBL6515272 0.80 TAS1R3 (0.42) TAS1R3TAS1R1ELANEMAPTANPEP
SCHEMBL6515278 0.80 TAS1R3 (0.42) TAS1R3TAS1R1ELANEMAPTANPEP
SCHEMBL6512117 0.79 CTSK (0.38) CYP2C9CYP2C19TAS1R3TAS1R1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005003103-A2 2, 4, 6-TRI-SUBSTITUTED 6-MEMBERED HETEROCYCLES AND THEIR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES ASTRAZENECA AB (SE) 2005-01-13 WO disclosed