SCHEMBL651778

SCHEMBL651778

Cc1ccccc1C[CH]c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.43
ALDH1A1 P00352 3/20 0.42
KMT2A Q03164 2/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.38
CTBP2 P56545 1/20 0.38
TSHR P16473 1/20 0.38
ACHE P22303 1/20 0.38
PTGS1 P23219 2/20 0.37
PTGS2 P35354 2/20 0.37
CHRM2 P08172 1/20 0.37
MAPT P10636 2/20 0.37
CYP2A6 P11509 1/20 0.37
KDM4E B2RXH2 1/20 0.37
P2RX7 Q99572 2/20 0.37
CCNB2 O95067 1/20 0.36
CDK1 P06493 1/20 0.36
CDK4 P11802 1/20 0.36
CCNB1 P14635 1/20 0.36
CCND1 P24385 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL397814 0.84 KDM4E (0.43) TAAR1ALDH1A1KMT2AHPGDPTGS1
SCHEMBL2250015 0.81 TRPA1 (0.47) ALDH1A1TSHRPTGS1PTGS2MAPT
SCHEMBL1932532 0.79 ALDH1A1 (0.55) TAAR1ALDH1A1KMT2APTGS1PTGS2
SCHEMBL1932534 0.79 ALDH1A1 (0.55) TAAR1ALDH1A1KMT2APTGS1PTGS2
SCHEMBL8368839 0.78 TSHR (0.46) TAAR1ALDH1A1KMT2AGAAHPGD
SCHEMBL19357314 0.77 CHRM5 (0.47) ALDH1A1KMT2AACHECCNB2CDK1
SCHEMBL3066574 0.76 NQO2 (0.42) ALDH1A1KMT2AGAAHPGDPTGS1
SCHEMBL1988589 0.75 TAAR1 (0.48) TAAR1ALDH1A1KMT2AGAAHPGD
SCHEMBL8397406 0.74 TAAR1 (0.45) TAAR1ALDH1A1KMT2ACYP2A6CYP2A13
SCHEMBL6085811 0.73 TAAR1 (0.46) TAAR1ALDH1A1KMT2AGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119667-B2 Carbonates of fenicol antibiotics SCHERING-PLOUGH ANIMAL HEALTH CORPORATION (US) 2012-02-21 US claimed
US-6479492-B1 TREATMENT OF INFLAMMATORY DISEASES IN A MAMMALIAN PATIENT ELAN PHARMACEUTICALS, INC. 2002-11-12 US claimed
CN-109232576-B 7-substituted desoxypeganone base and preparation method and application thereof 信阳师范学院 2020-07-17 CN disclosed
WO-2013187978-A1 DOUBLE-LIVER-TARGETING PHOSPHORAMIDATE AND PHOSPHONOAMIDATE PRODRUGS NANJING MOLECULAR RESEARCH, INC. (CN) 2013-12-19 WO disclosed
US-7538215-B2 Compounds which inhibit leukocyte adhesion mediated by VLA-4 ELAN PHARMACEUTICALS, INC. (US) 2009-05-26 US disclosed
EP-1144384-B1 COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARM INC (US) 2007-10-31 EP disclosed
US-20050261293-A1 Compounds which inhibit leukocyte adhesion mediated by VLA-4 WYETH 2005-11-24 US disclosed
US-6903088-B2 Compounds which inhibit leukocyte adhesion mediated by VLA-4 ELAN PHARMACEUTICALS, INC. (US) 2005-06-07 US disclosed
US-6479492-B1 TREATMENT OF INFLAMMATORY DISEASES IN A MAMMALIAN PATIENT ELAN PHARMACEUTICALS, INC. 2002-11-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050261293-A1 Compounds which inhibit leukocyte adhesion mediated by VLA-4 VCAM1, ICAM1, CD4 TAAR1 3380/4885ALDH1A1 322/4885KMT2A 1871/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.