SCHEMBL6519845

SCHEMBL6519845

C=CCN1CCc2ccccc2C1.Cc1ccc(S(=O)(=O)O)cc1

nearest known ligand 0.57

Known targets — ChEMBL curated mechanism

ABL1BMXBRAFBTKCHRNA4CHRNB2CSNK1EEGFRERBB2F10FLT1FLT3FLT4IGF1RINSRITKJAK3KDRKITOPRM1PARP1PARP2PDGFRBPIK3CDRAF1RETSLC18A2TECTXKdacAdacBdacCftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.53
MEN1 O00255 5/20 0.53
ALDH1A1 P00352 3/20 0.51
KDM4E B2RXH2 2/20 0.51
PKM P14618 1/20 0.51
TSHR P16473 1/20 0.51
USP2 O75604 1/20 0.49
TAAR1 Q96RJ0 1/20 0.49
OPRK1 P41145 1/20 0.46
LMNA P02545 2/20 0.44
GAA P10253 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NOD1 Q9Y239 1/20 0.44
HTT P42858 2/20 0.43
HPGD P15428 1/20 0.43
POLB P06746 1/20 0.43
NR4A1 P22736 1/20 0.43
ESR2 Q92731 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ADRA1D P25100 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6521329 0.90 HTR7 (0.52) KMT2AMEN1ALDH1A1KDM4EPKM
SCHEMBL6527411 0.82 USP2 (0.54) KMT2AMEN1ALDH1A1KDM4EPKM
SCHEMBL3957205 0.81 ADRA1D (0.62) ALDH1A1KDM4EADRA1DADRA1AADRA1B
SCHEMBL6521515 0.81 HTR7 (0.54) KMT2AMEN1ALDH1A1KDM4EPKM
Acetic Acid SCHEMBL6519592 0.80 HDAC3 (0.52) KMT2AMEN1KDM4EPOLBADRA1D
Bromide SCHEMBL6521671 0.80 ADRA1D (0.61) ALDH1A1KDM4ELMNAADRA1DADRA1A
SCHEMBL6524885 0.79 MAOA (0.61) KMT2AMEN1ALDH1A1KDM4EPKM
SCHEMBL8779551 0.79 HTR7 (0.55) KMT2AMEN1ALDH1A1KDM4EPKM
SCHEMBL28743871 0.77 MEN1 (0.48) KMT2AMEN1ALDH1A1KDM4EPKM
SCHEMBL20891206 0.74 ADRA1D (0.42) KMT2AMEN1ALDH1A1GAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274056-B1 BLEACHING AGENT COMPRISING CATIONIC 3,4-DIHYDROISOCHINOLINIUM DERIVATIVES, SPECIFIC ALKANOLAMINES AND HYDROGEN PEROXYDE HENKEL AG & CO KGAA (DE) 2012-10-03 EP claimed
US-20110056508-A1 BLEACHING AGENT COMPRISING CATIONIC 3,4-DIHYDROISOQUINOLINE DERIVATIVES, SPECIAL ALKANOL AMINES AND HYDROGEN PEROXIDE GROSS WIBKE 2011-03-10 US claimed
US-20110056508-A1 BLEACHING AGENT COMPRISING CATIONIC 3,4-DIHYDROISOQUINOLINE DERIVATIVES, SPECIAL ALKANOL AMINES AND HYDROGEN PEROXIDE GROSS WIBKE 2011-03-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110056508-A1 BLEACHING AGENT COMPRISING CATIONIC 3,4-DIHYDROISOQUINOLINE DERIVATIVES, SPECIAL ALKANOL AMINES AND HYDROGEN PEROXIDE KRT18, H1-3, H1-2 KMT2A 217/4885MEN1 4466/4885ALDH1A1 152/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.