SCHEMBL6521387

SCHEMBL6521387

Cc1c(-c2cccc(Cl)c2)nc2ccc(-c3ccc(F)c(CO)c3F)cn12

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 2/20 0.51
TRPA1 O75762 6/20 0.43
NR1H4 Q96RI1 2/20 0.43
ATM Q13315 4/20 0.43
SLC2A1 P11166 2/20 0.40
MAPT P10636 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
PSMD14 O00487 1/20 0.37
CASP3 P42574 1/20 0.37
SENP8 Q96LD8 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6521811 0.91 TRPA1 (0.42) NR4A2TRPA1NR1H4ATMSLC2A1
SCHEMBL6520541 0.89 NR4A2 (0.61) NR4A2NR1H4SLC2A1MAPTCYP11B1
SCHEMBL6519571 0.89 NR4A2 (0.50) NR4A2NR1H4ATMSLC2A1MAPT
SCHEMBL6527443 0.82 NR4A2 (0.47) NR4A2NR1H4ATMSLC2A1MAPT
SCHEMBL3431442 0.81 NR4A2 (0.47) NR4A2NR1H4SLC2A1MAPT
SCHEMBL3431629 0.80 NR4A2 (0.46) NR4A2NR1H4SLC2A1
SCHEMBL6524183 0.79 DHODH (0.44) NR1H4SLC2A1MAPTNPC1RAB9A
SCHEMBL16208077 0.79 NR4A2 (0.65) NR4A2SLC2A1MAPT
SCHEMBL218112 0.76 SOS1 (0.44) TRPA1NR1H4ATMSLC2A1MAPT
SCHEMBL6524569 0.76 DHODH (0.43) NR4A2TRPA1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262769-B1 POLYSUBSTITUTED 2-ARYL-6-PHENYL-IMIDAZO[1,2-A]PYRIDINE DERIVATIVES, AND PREPARATION AND THERAPEUTIC USE THEREOF SANOFI SA (FR) 2014-11-05 EP claimed
EP-2262769-B1 POLYSUBSTITUTED 2-ARYL-6-PHENYL-IMIDAZO[1,2-A]PYRIDINE DERIVATIVES, AND PREPARATION AND THERAPEUTIC USE THEREOF SANOFI SA (FR) 2014-11-05 EP disclosed
US-20110065745-A1 POLYSUBSTITUTED 2-ARYL-6-PHENYLIMIDAZO[1,2-A]PYRIDINE DERIVATIVES, AND PREPARATION AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-03-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110065745-A1 POLYSUBSTITUTED 2-ARYL-6-PHENYLIMIDAZO[1,2-A]PYRIDINE DERIVATIVES, AND PREPARATION AND THERAPEUTIC USE THEREOF JAK2, ABL1, REN NR4A2 1394/4885TRPA1 3023/4885NR1H4 393/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.