SCHEMBL6525004

SCHEMBL6525004

O=C1c2ccccc2C(=O)N1OC1COC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.42
ALDH1A1 P00352 7/20 0.40
MAPT P10636 5/20 0.40
KMT2A Q03164 4/20 0.40
HPGD P15428 4/20 0.40
KDM4E B2RXH2 3/20 0.40
MEN1 O00255 3/20 0.37
CYP1A2 P05177 3/20 0.37
CYP2C9 P11712 2/20 0.37
VDR P11473 1/20 0.37
NSD2 O96028 1/20 0.36
G6PD P11413 1/20 0.36
CCR6 P51684 1/20 0.36
PKM P14618 1/20 0.35
ALOX15 P16050 1/20 0.35
ALOX12 P18054 1/20 0.35
MC4R P32245 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CYP2C19 P33261 2/20 0.35
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4864756 0.86 CYP1A2 (0.38) GAAALDH1A1MAPTKMT2AHPGD
SCHEMBL30728974 0.82 GAA (0.46) GAAALDH1A1MAPTKMT2AHPGD
SCHEMBL30137583 0.82 GAA (0.40) GAAALDH1A1MAPTKMT2AHPGD
SCHEMBL4863817 0.82 GAA (0.40) GAAALDH1A1MAPTKMT2AHPGD
SCHEMBL4856718 0.82 LMNA (0.37) GAAALDH1A1MAPTKMT2AHPGD
SCHEMBL2565587 0.80 KMT2A (0.39) GAAALDH1A1MAPTKMT2AHPGD
SCHEMBL24130978 0.79 ALDH1A1 (0.43) GAAALDH1A1MAPTKMT2AHPGD
SCHEMBL9388231 0.79 GAA (0.43) GAAALDH1A1MAPTKMT2AHPGD
SCHEMBL30002131 0.79 ALDH1A1 (0.47) GAAALDH1A1MAPTKMT2AHPGD
SCHEMBL2077862 0.79 ALDH1A1 (0.47) GAAALDH1A1MAPTKMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 42 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12486274-B2 Substituted pyrazolo-pyrimidines and uses thereof Verge Analytics, Inc. (US) 2025-12-02 US disclosed
EP-4647127-A2 COMPOUNDS FOR THE TREATMENT OF KINASE-DEPENDENT DISORDERS Exelixis, Inc. (US) 2025-11-12 EP disclosed
EP-3743070-B1 COMPOUNDS FOR THE TREATMENT OF KINASE-DEPENDENT DISORDERS EXELIXIS INC (US) 2025-07-23 EP disclosed
CN-115209952-B Substituted pyrazolopyrimidines and use thereof 维基分析有限公司 2025-05-30 CN disclosed
CN-117820226-A Compounds for the treatment of kinase dependent disorders 埃克塞里艾克西斯公司 2024-04-05 CN disclosed
CN-117624045-A Compounds for the treatment of kinase dependent disorders 埃克塞里艾克西斯公司 2024-03-01 CN disclosed
CN-117603138-A Compounds for the treatment of kinase dependent disorders 埃克塞里艾克西斯公司 2024-02-27 CN disclosed
US-20240043414-A1 Compounds for the Treatment of Kinase-Dependent Disorders EXELIXIS, INC. 2024-02-08 US disclosed
CN-117402114-A Compounds for the treatment of kinase dependent disorders 埃克塞里艾克西斯公司 2024-01-16 CN disclosed
CN-111757735-B Compounds for the treatment of kinase dependent disorders 埃克塞里艾克西斯公司 2023-09-22 CN disclosed
US-8410264-B2 Heterocyclic oxime compounds NOVARTIS AG (CH) 2013-04-02 US disclosed
US-20120302570-A1 HETEROCYCLIC OXIME COMPOUNDS NOVARTIS AG (CH) 2012-11-29 US disclosed
US-20120302570-A1 HETEROCYCLIC OXIME COMPOUNDS NOVARTIS AG (CH) 2012-11-29 US disclosed
US-20120302570-A1 HETEROCYCLIC OXIME COMPOUNDS NOVARTIS AG (CH) 2012-11-29 US disclosed
EP-2467383-A1 HETEROCYCLIC OXIME COMPOUNDS Novartis AG (CH) 2012-06-27 EP disclosed
US-20110065708-A1 HETEROCYCLIC OXIME COMPOUNDS NOVARTIS AG (CH) 2011-03-17 US disclosed
US-20110065708-A1 HETEROCYCLIC OXIME COMPOUNDS NOVARTIS AG (CH) 2011-03-17 US disclosed
US-20110065708-A1 HETEROCYCLIC OXIME COMPOUNDS NOVARTIS AG (CH) 2011-03-17 US disclosed
WO-2011020861-A1 HETEROCYCLIC OXIME COMPOUNDS NOVARTIS AG (CH) 2011-02-24 WO disclosed
WO-2011020861-A1 HETEROCYCLIC OXIME COMPOUNDS NOVARTIS AG (CH) 2011-02-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12486274-B2 Substituted pyrazolo-pyrimidines and uses thereof PIKFYVE, PIP4K2B, PIP4K2C GAA 792/4885ALDH1A1 4827/4885MAPT 770/4885
US-20110065708-A1 HETEROCYCLIC OXIME COMPOUNDS MET, ERBB2, TIE1 GAA 2312/4885ALDH1A1 430/4885MAPT 2873/4885
US-20120302570-A1 HETEROCYCLIC OXIME COMPOUNDS MET, ERBB2, TIE1 GAA 2312/4885ALDH1A1 430/4885MAPT 2873/4885
US-20240043414-A1 Compounds for the Treatment of Kinase-Dependent Disorders ERBB2, MAP3K6, MAP3K1 GAA 535/4885ALDH1A1 3310/4885MAPT 1513/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.