SCHEMBL6528259

SCHEMBL6528259

CS(=O)(=O)NS(C)(=O)=O.Fc1ccccc1Cn1cnc2cnc(C(F)(F)F)nc21

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 9/20 0.56
PDE4B Q07343 9/20 0.56
PDE4C Q08493 9/20 0.56
PDE4D Q08499 9/20 0.56
PDE5A O76074 3/20 0.56
PDE1A P54750 3/20 0.56
PDE1B Q01064 3/20 0.56
PDE1C Q14123 3/20 0.56
PDE3B Q13370 3/20 0.48
PDE3A Q14432 3/20 0.48
HDAC6 Q9UBN7 1/20 0.43
YTHDC1 Q96MU7 2/20 0.40
LMNA P02545 1/20 0.39
CNR2 P34972 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
DDR1 Q08345 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dimethylamine SCHEMBL4532702 0.89 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL6528258 0.74 PDE4A (0.63) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL9738442 0.74 PDE4A (0.56) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL9738484 0.72 FGFR1 (0.49) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL4460149 0.72 PDE4A (0.73) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL185397 0.72 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL29798952 0.72 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL9738952 0.72 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL11014177 0.72 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL3141400 0.71 PDE4A (0.82) PDE4APDE4BPDE4CPDE4DPDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1551837-A1 PHOSPHODIESTERASE 4 INHIBITORS Memory Pharmaceutical Corporation (US) 2005-07-13 EP claimed
WO-2004014911-A1 PHOSPHODIESTERASE 4 INHIBITORS MEMORY PHARMACEUTICALS CORPORATION (US) 2004-02-19 WO claimed