SCHEMBL6529486

SCHEMBL6529486

NC(=O)Nc1sc(C(=O)NO)cc1C(=O)NO

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 13/20 0.46
MAP4K4 O95819 1/20 0.46
IKBKB O14920 4/20 0.43
JAK2 O60674 2/20 0.43
JAK3 P52333 1/20 0.43
HDAC6 Q9UBN7 4/20 0.41
HDAC3 O15379 3/20 0.41
HDAC4 P56524 3/20 0.41
HDAC1 Q13547 3/20 0.41
HDAC7 Q8WUI4 3/20 0.41
HDAC2 Q92769 3/20 0.41
HDAC10 Q969S8 3/20 0.41
HDAC11 Q96DB2 3/20 0.41
HDAC8 Q9BY41 3/20 0.41
HDAC9 Q9UKV0 3/20 0.41
HDAC5 Q9UQL6 3/20 0.41
MEN1 O00255 1/20 0.41
EIF2AK2 P19525 1/20 0.41
KMT2A Q03164 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6532445 0.93 IKBKB (0.44) CHEK1MAP4K4IKBKBJAK2JAK3
SCHEMBL6507152 0.78 IKBKB (0.57) CHEK1IKBKBJAK2JAK3HDAC6
SCHEMBL6505865 0.75 IKBKB (0.58) CHEK1MAP4K4IKBKBJAK2JAK3
SCHEMBL6507636 0.72 IKBKB (0.51) CHEK1IKBKBJAK2JAK3HDAC6
SCHEMBL6528389 0.71 IKBKB (0.50) CHEK1IKBKBHDAC6HDAC3HDAC4
SCHEMBL6505484 0.71 CHEK1 (0.55) CHEK1IKBKBJAK2JAK3HDAC6
SCHEMBL13667938 0.71 CHEK1 (0.59) CHEK1MAP4K4IKBKBJAK2JAK3
SCHEMBL491042 0.69 IKBKB (0.55) CHEK1IKBKBJAK2JAK3HDAC6
SCHEMBL6506758 0.69 IKBKB (0.50) CHEK1IKBKBJAK2JAK3MEN1
SCHEMBL6514837 0.68 CHEK1 (0.47) CHEK1IKBKBJAK2JAK3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005105777-A1 SUBSTITUTED THIOPHENE AMIDE COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA & UPJOHN COMPANY LLC (US) 2005-11-10 WO disclosed