SCHEMBL6530703

SCHEMBL6530703

NC(=O)Nc1sc(C(=O)NCc2ccccc2Cl)cc1C(N)=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 2/20 0.51
HDAC1 Q13547 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
MAPT P10636 3/20 0.48
POLB P06746 1/20 0.48
MAPK8 P45983 1/20 0.48
JAK2 O60674 1/20 0.47
JAK3 P52333 1/20 0.47
TP53 P04637 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
BACE1 P56817 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
LMNA P02545 1/20 0.45
CNR1 P21554 1/20 0.45
CNR2 P34972 1/20 0.45
ALDH1A1 P00352 2/20 0.44
KMT2A Q03164 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6511844 0.81 CYP2C19 (0.51) IKBKBMAPTMAPK8JAK2JAK3
SCHEMBL6514861 0.81 DYRK1A (0.52) IKBKBMAPTMAPK8JAK2JAK3
SCHEMBL23474255 0.73 TP53 (0.54) HDAC1HDAC6MAPTPOLBTP53
SCHEMBL10321814 0.73 SMN1; SMN2 (0.60) MAPTTP53NPC1RAB9ASMN1; SMN2
SCHEMBL23511435 0.72 HDAC1 (0.56) HDAC1HDAC6MAPTPOLBTP53
SCHEMBL6506758 0.72 IKBKB (0.50) IKBKBMAPTJAK2JAK3TP53
SCHEMBL625881 0.72 NPC1 (0.72) POLBTP53NPC1RAB9ASMN1; SMN2
SCHEMBL6507152 0.72 IKBKB (0.57) IKBKBHDAC6JAK2JAK3TDP1
SCHEMBL6506008 0.72 IKBKB (0.56) IKBKBHDAC6POLBJAK2JAK3
SCHEMBL23511678 0.71 HDAC1 (0.51) HDAC1HDAC6MAPTPOLBTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005105777-A1 SUBSTITUTED THIOPHENE AMIDE COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA & UPJOHN COMPANY LLC (US) 2005-11-10 WO disclosed