SCHEMBL6506008

SCHEMBL6506008

NC(=O)Nc1sc(NC(=O)c2ccccc2Cl)cc1C(N)=O

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 7/20 0.56
JAK2 O60674 2/20 0.52
JAK3 P52333 1/20 0.52
RAB9A P51151 2/20 0.48
CFTR P13569 1/20 0.48
NPC1 O15118 1/20 0.48
MEN1 O00255 1/20 0.47
EIF2AK2 P19525 1/20 0.47
KMT2A Q03164 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
CYP1A2 P05177 1/20 0.47
HPGD P15428 1/20 0.47
CYP2C19 P33261 1/20 0.47
CHEK1 O14757 1/20 0.45
POLB P06746 1/20 0.44
KCNK3 O14649 1/20 0.43
KCNK9 Q9NPC2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6504891 0.85 IKBKB (0.57) IKBKBJAK2JAK3RAB9ANPC1
SCHEMBL6507659 0.82 IKBKB (0.53) IKBKBJAK2JAK3RAB9ANPC1
SCHEMBL6508136 0.82 IKBKB (0.60) IKBKBJAK2JAK3MEN1EIF2AK2
SCHEMBL6503091 0.82 IKBKB (0.50) IKBKBJAK2JAK3MEN1EIF2AK2
SCHEMBL6507070 0.82 IKBKB (0.46) IKBKBJAK2JAK3MEN1EIF2AK2
SCHEMBL6505282 0.81 MAPT (0.55) IKBKBJAK2JAK3RAB9ANPC1
SCHEMBL6530279 0.80 IKBKB (0.48) IKBKBJAK2JAK3RAB9ANPC1
SCHEMBL6506340 0.80 FLT3 (0.51) IKBKBJAK2JAK3RAB9ANPC1
SCHEMBL6509362 0.78 OGG1 (0.54) RAB9ANPC1MEN1KMT2AHDAC6
SCHEMBL7004222 0.78 JAK2 (0.69) IKBKBJAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005105777-A1 SUBSTITUTED THIOPHENE AMIDE COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA & UPJOHN COMPANY LLC (US) 2005-11-10 WO disclosed