SCHEMBL6531003

SCHEMBL6531003

COc1ccc(-c2nc(Cl)nc(Nc3cccc(F)c3)n2)cc1

nearest known ligand 0.63

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 5/20 0.63
APP P05067 2/20 0.57
MAPT P10636 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
RORC P51449 8/20 0.52
ABCG2 Q9UNQ0 2/20 0.48
DHFR P00374 1/20 0.48
PIK3CA P42336 1/20 0.46
PIK3CG P48736 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22123529 0.85 ABCG2 (0.58) APPMAPTSMN1; SMN2ABCG2
SCHEMBL8298690 0.81 APP (0.54) CHRNA7APPMAPTSMN1; SMN2
SCHEMBL6529150 0.81 CHRNA7 (0.61) CHRNA7APPMAPTSMN1; SMN2
SCHEMBL2874930 0.79 NFKB1 (0.65) CHRNA7APPMAPTSMN1; SMN2
SCHEMBL28929970 0.77 CHRNA7 (1.00) CHRNA7APPMAPTSMN1; SMN2
SCHEMBL1594413 0.77 ADORA2A (0.57) CHRNA7APPMAPTSMN1; SMN2ABCG2
SCHEMBL1592702 0.75 ABCG2 (0.57) CHRNA7APPMAPTSMN1; SMN2ABCG2
SCHEMBL30933621 0.75 TXN (0.46) CHRNA7APPMAPTSMN1; SMN2RORC
SCHEMBL6530084 0.75 RORC (0.45) CHRNA7RORCABCG2DHFR
SCHEMBL6530078 0.75 RORC (0.45) CHRNA7RORCABCG2DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005003103-A2 2, 4, 6-TRI-SUBSTITUTED 6-MEMBERED HETEROCYCLES AND THEIR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES ASTRAZENECA AB (SE) 2005-01-13 WO disclosed
WO-2005003103-A2 2, 4, 6-TRI-SUBSTITUTED 6-MEMBERED HETEROCYCLES AND THEIR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES ASTRAZENECA AB (SE) 2005-01-13 WO disclosed