SCHEMBL653335

SCHEMBL653335

CC(C)(NC(=O)c1cc2[nH]nc(NC(=O)c3ccccc3N)c2o1)c1ccccc1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FADS1 O60427 3/20 0.36
P2RX1 P51575 1/20 0.35
SMN1; SMN2 Q16637 4/20 0.34
PTGS1 P23219 2/20 0.34
ALDH1A1 P00352 2/20 0.34
GLA P06280 1/20 0.34
AURKA O14965 1/20 0.34
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
GAA P10253 2/20 0.33
INSR P06213 1/20 0.33
IGF1R P08069 1/20 0.33
ALK Q9UM73 1/20 0.33
HDAC6 Q9UBN7 2/20 0.33
MAPK1 P28482 1/20 0.33
KDR P35968 1/20 0.33
GCK P35557 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL653354 0.88 RXFP1 (0.38) SMN1; SMN2ALDH1A1GLANPC1RAB9A
SCHEMBL655164 0.88 AURKA (0.42) FADS1P2RX1SMN1; SMN2PTGS1ALDH1A1
SCHEMBL4084047 0.87 AURKA (0.42) AURKAHDAC6HDAC3HDAC1HDAC2
SCHEMBL652599 0.87 MEN1 (0.41) P2RX1SMN1; SMN2ALDH1A1NPC1RAB9A
SCHEMBL4082088 0.85 SMN1; SMN2 (0.41) SMN1; SMN2ALDH1A1NPC1RAB9AMAPK1
SCHEMBL653322 0.85 ALK (0.54) AURKAINSRIGF1RALKKDR
SCHEMBL4091695 0.84 MAPK1 (0.45) SMN1; SMN2ALDH1A1NPC1RAB9AGAA
SCHEMBL4083477 0.84 AURKA (0.42) SMN1; SMN2ALDH1A1GLAAURKANPC1
SCHEMBL13850096 0.84 AURKA (0.39) AURKAINSRIGF1RALKHDAC6
SCHEMBL652592 0.84 PPARG (0.35) SMN1; SMN2ALDH1A1GLAAURKANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119641-B2 1H-furo[3,2-C]pyrazole compounds useful as kinase inhibitors NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2012-02-21 US disclosed