SCHEMBL6534342

SCHEMBL6534342

Clc1cc(-c2cc3ccccc3s2)nc2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
RXFP1 Q9HBX9 2/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
GLA P06280 1/20 0.45
GAA P10253 1/20 0.45
PPARG P37231 1/20 0.45
NCOA2 Q15596 1/20 0.45
NCOA1 Q15788 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
ACP1 P24666 1/20 0.43
CYP19A1 P11511 1/20 0.43
NQO1 P15559 1/20 0.42
NQO2 P16083 1/20 0.42
KDM1A O60341 2/20 0.42
APP P05067 2/20 0.41
PGK1 P00558 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6694034 0.85 CYP19A1 (0.41) ACP1CYP19A1NQO1NQO2KDM1A
SCHEMBL13220280 0.80 CYP19A1 (0.48) ALDH1A1CYP19A1NQO1NQO2KDM1A
SCHEMBL29263263 0.78 BACE1 (0.54) MEN1KMT2ARXFP1KDM4EALDH1A1
SCHEMBL31023423 0.78 BACE1 (0.54) MEN1KMT2ARXFP1KDM4EALDH1A1
SCHEMBL2208526 0.76 RAB9A (0.54) MEN1KMT2AKDM4EALDH1A1SMN1; SMN2
SCHEMBL4492064 0.76 TERT (0.42) MEN1KMT2AALDH1A1SMN1; SMN2NQO1
SCHEMBL31038115 0.76 RAB9A (0.54) MEN1KMT2AKDM4EALDH1A1SMN1; SMN2
SCHEMBL29793367 0.73 ACHE (0.61) MEN1KMT2AKDM4EALDH1A1LMNA
SCHEMBL785473 0.73 ACHE (0.61) MEN1KMT2AKDM4EALDH1A1LMNA
SCHEMBL12383603 0.73 NQO1 (0.45) CYP19A1NQO1NQO2KDM1AAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1088818-B1 Quinolin-4-yl derivatives HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed
US-6440995-B1 NMDA-RECEPTOR SUBTYPE SELECTIVE BLOCKERS HOFFMAN-LA ROCHE INC. 2002-08-27 US disclosed
EP-1088818-A1 Quinolin-4-yl derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-04-04 EP disclosed