SCHEMBL6534835

SCHEMBL6534835

CC(C)(C)OC(=O)CC(N)(CN)CC(=O)OC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.35
CYP2D6 P10635 1/20 0.32
DGAT1 O75907 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
CA12 O43570 1/20 0.30
CA2 P00918 1/20 0.30
CA14 Q9ULX7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6535010 0.98 KDM4E (0.39) KDM4ECYP2D6DGAT1HDAC3HDAC1
SCHEMBL29550018 0.83 KDM4E (0.35) KDM4ECYP2D6DGAT1HDAC3HDAC1
SCHEMBL1951896 0.80 KDM4E (0.52) KDM4ECYP2D6DGAT1HDAC3HDAC1
SCHEMBL7826803 0.79 DGAT1 (0.34) KDM4ECYP2D6DGAT1HDAC3HDAC1
SCHEMBL31238586 0.79 HDAC3 (0.37) CYP2D6DGAT1HDAC3HDAC1HDAC2
SCHEMBL12348352 0.79 STING1 (0.34) CYP2D6HDAC3HDAC1HDAC2HDAC8
SCHEMBL28832570 0.77 DGAT1 (0.33) CYP2D6DGAT1HDAC3HDAC1HDAC2
SCHEMBL27443265 0.76 CYP2D6 (0.33) CYP2D6DGAT1HDAC3HDAC1HDAC2
SCHEMBL1952236 0.75 KDM4E (0.33) KDM4ECYP2D6DGAT1CA12CA2
SCHEMBL189917 0.74 GGT1 (0.41) KDM4ECYP2D6DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0941120-A4 BRANCHED PEPTIDE LINKERS BRISTOL MYERS SQUIBB CO (US) 2004-08-18 EP disclosed
EP-0941120-A1 BRANCHED PEPTIDE LINKERS BRISTOL-MYERS SQUIBB COMPANY (US) 1999-09-15 EP disclosed
WO-1998019705-A1 BRANCHED PEPTIDE LINKERS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-14 WO disclosed