SCHEMBL6535408

SCHEMBL6535408

Oc1ccccc1C(COc1ccccc1)CSCC(COc1ccccc1)c1ccccc1O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.44
SCN4A P35499 2/20 0.40
TSHR P16473 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MAOA P21397 1/20 0.38
PTGS1 P23219 1/20 0.38
MTNR1A P48039 3/20 0.37
MTNR1B P49286 3/20 0.37
CYP2D6 P10635 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
ADRB2 P07550 1/20 0.37
ADRB1 P08588 1/20 0.37
ADRB3 P13945 1/20 0.37
GABRA1 P14867 1/20 0.37
GABRB2 P47870 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
RECQL P46063 1/20 0.36
BACE1 P56817 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6535124 0.79 TSHR (0.44) LMNATSHRKMT2AGABRA1GABRB2
SCHEMBL7994693 0.78 MTNR1A (0.43) LMNATSHRKMT2AHSD17B10PTGS1
SCHEMBL9854863 0.76 TSHR (0.58) LMNASCN4ATSHRKMT2AMAOA
SCHEMBL8002064 0.76 POLB (0.44) TSHRPTGS1MTNR1AMTNR1BGABRA1
SCHEMBL28814512 0.74 LTA4H (0.43) LMNATSHRMAOAADRB2ADRB1
SCHEMBL6534959 0.72 TSHR (0.48) LMNATSHRHSD17B10L3MBTL1GABRA1
SCHEMBL15079881 0.72 LTA4H (0.49) LMNACYP2D6L3MBTL1ADRB2ADRB1
SCHEMBL7998182 0.70 TSHR (0.38) TSHRGABRA1GABRB2
SCHEMBL6534892 0.70 TSHR (0.46) LMNATSHRKMT2AHSD17B10GABRA1
SCHEMBL7996412 0.70 CYSLTR2 (0.47) TSHRCYP2D6GABRA1GABRB2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0958275-A4 SELECTIVE INHIBITORS OF PROSTAGLANDIN ENDOPEROXIDE SYNTHASE-2 UNIV VANDERBILT (US) 2004-12-01 EP disclosed
US-6284918-B1 ENZYME INHIBITORS VANDERBILT UNIVERSITY 2001-09-04 US disclosed
EP-0958275-A1 SELECTIVE INHIBITORS OF PROSTAGLANDIN ENDOPEROXIDE SYNTHASE-2 VANDERBILT UNIVERSITY (US) 1999-11-24 EP disclosed
US-5973191-A AN ACETOXYPHENYLALKYL SULFIDE, SALT OR HYDRATE VANDERBILT UNIVERSITY (US) 1999-10-26 US disclosed
WO-1998029382-A1 SELECTIVE INHIBITORS OF PROSTAGLANDIN ENDOPEROXIDE SYNTHASE-2 VANDERBILT UNIVERSITY (US) 1998-07-09 WO disclosed