SCHEMBL6535966

SCHEMBL6535966

COC(=O)c1ccc(-c2cccc(OC)c2OC)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.50
ADORA2A P29274 2/20 0.50
ADORA2B P29275 2/20 0.50
PTPRC P08575 1/20 0.50
PTPRF P10586 1/20 0.50
PTPN1 P18031 1/20 0.50
CDC25B P30305 1/20 0.50
PTGS1 P23219 1/20 0.49
EGFR P00533 1/20 0.49
KDM4E B2RXH2 1/20 0.48
HSD17B10 Q99714 1/20 0.48
STIM1 Q13586 2/20 0.47
ORAI1 Q96D31 2/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
TSHR P16473 1/20 0.46
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45
FFAR4 Q5NUL3 1/20 0.45
ROCK2 O75116 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2042640 0.86 STIM1 (0.57) ADORA3ADORA2AADORA2BKDM4EHSD17B10
SCHEMBL6773146 0.86 KDM4E (0.56) EGFRKDM4EHSD17B10CA1CA2
SCHEMBL29868499 0.86 KDM4E (0.56) EGFRKDM4EHSD17B10CA1CA2
SCHEMBL2050621 0.85 EGFR (0.56) PTPRCPTPRFPTPN1CDC25BPTGS1
SCHEMBL29788043 0.85 EGFR (0.56) PTPRCPTPRFPTPN1CDC25BPTGS1
SCHEMBL12844713 0.85 ERN1 (0.52) ADORA3ADORA2AADORA2BSTIM1ORAI1
SCHEMBL7359469 0.84 STIM1 (0.47) ADORA3ADORA2AADORA2BKDM4EHSD17B10
SCHEMBL27499555 0.83 LMNA (0.58) ADORA3ADORA2AADORA2BPTGS1KDM4E
SCHEMBL28092583 0.78 MGAM (0.54) ADORA3ADORA2AADORA2BKDM4EHSD17B10
SCHEMBL4778742 0.78 ALDH1A1 (0.56) ADORA3ADORA2AADORA2BKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1425015-A4 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL MYERS SQUIBB CO (US) 2004-12-15 EP disclosed
EP-1425015-A2 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-06-09 EP disclosed
WO-2003015715-A2 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-02-27 WO disclosed