SCHEMBL6773146

SCHEMBL6773146

COC(=O)c1ccc(-c2ccc(OC)c(OC)c2OC)cc1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.56
HSD17B10 Q99714 1/20 0.56
EGFR P00533 2/20 0.50
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
MAPT P10636 3/20 0.48
ERN1 O75460 2/20 0.47
CYP3A4 P08684 1/20 0.47
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
TDP1 Q9NUW8 1/20 0.46
CA12 O43570 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29868499 1.00 KDM4E (0.56) KDM4EHSD17B10EGFRCA1CA2
SCHEMBL6535966 0.86 ADORA3 (0.50) KDM4EHSD17B10EGFRCA1CA2
SCHEMBL6769062 0.85 ERN1 (0.48) MAPTERN1KMT2AMEN1
SCHEMBL2044179 0.85 CA1 (0.51) EGFRCA1CA2MAPTERN1
SCHEMBL29788180 0.85 CA1 (0.51) EGFRCA1CA2MAPTERN1
SCHEMBL1617752 0.82 ERN1 (0.51) KDM4EHSD17B10CA1CA2MAPT
SCHEMBL31238859 0.80 MAPT (0.58) KDM4EEGFRCA1CA2MAPT
SCHEMBL10459227 0.79 KDM4E (0.46) KDM4EHSD17B10EGFRCA1CA2
SCHEMBL2050621 0.77 EGFR (0.56) EGFRCA1CA2MAPT
SCHEMBL21182648 0.77 EGFR (0.56) KDM4EEGFRCA1CA2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6673814-B2 CONTROLLED-RELEASE BY IMPLANTABLE DEVICES, DELIVERY PUMPS, WAFERS, AND BIODEGRADABLE POLYMERS EMORY UNIVERSITY 2004-01-06 US disclosed
US-20020137762-A1 Delivery systems and methods for noscapine and noscapine derivatives, useful as anticancer agents EMORY UNIVERSITY 2002-09-26 US disclosed
US-6376516-B1 FOR TREATING NEOPLASTIC CANCERS INCLUDING COLON, LUNG, BRAIN, OVARIAN, PROSTATE, BREAST, AND BLADDER CANCER AND LEUKEMIA; LOW TOXICITY EMORY UNIVERSITY 2002-04-23 US disclosed
WO-1999008528-A1 NOSCAPINE DERIVATIVES, USEFUL AS ANTICANCER AGENTS EMORY UNIVERSITY (US) 1999-02-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020137762-A1 Delivery systems and methods for noscapine and noscapine derivatives, useful as anticancer agents NOS1, NOS2, HCCS KDM4E 2873/4885HSD17B10 1421/4885EGFR 1408/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.