SCHEMBL6536683

SCHEMBL6536683

CCOC(=O)CNS(=O)(=O)c1ccc2c(c1)C(=O)C(=O)N2

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
CASP3 P42574 5/20 0.45
APEX1 P27695 1/20 0.44
HPGD P15428 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
PDPK1 O15530 1/20 0.43
CASP7 P55210 2/20 0.43
SYK P43405 2/20 0.42
FCER2 P06734 1/20 0.42
PKM P14618 1/20 0.42
CASP1 P29466 1/20 0.42
CASP9 P55211 1/20 0.42
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6535147 0.79 CASP3 (0.73) CASP3CASP7CASP1CASP9
SCHEMBL1091461 0.78 CA12 (0.55) ALDH1A1CA12CA1CA2CA9
SCHEMBL257480 0.78 ALDH1A1 (0.67) ALDH1A1HPGDPKMKMT2A
SCHEMBL14111831 0.75 ALDH1A1 (0.67) ALDH1A1CA12CA1CA2CA9
SCHEMBL12273071 0.75 TGM2 (0.56) ALDH1A1
SCHEMBL13917758 0.74 ALDH1A1 (0.62) ALDH1A1HPGDPKMKMT2A
SCHEMBL13065421 0.74 ALDH1A1 (0.55) ALDH1A1HPGDPKM
SCHEMBL10420167 0.74 GAA (0.65) ALDH1A1NPSR1PKMKMT2A
SCHEMBL15595362 0.74 HTT (0.56) ALDH1A1NPSR1KMT2A
SCHEMBL5894519 0.73 CA12 (0.63) ALDH1A1CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403792-B1 INHIBIT PRODUCTION OF CASPASE 3 AND 7 IN MAMMALS SMITHKLINE BEECHAM CORPORATION 2002-06-11 US claimed
EP-1242081-A4 CASPASES AND APOPTOSIS SMITHKLINE BEECHAM CORP (US) 2004-07-21 EP disclosed
EP-1242081-A1 CASPASES AND APOPTOSIS SmithKline Beecham Corporation (US) 2002-09-25 EP disclosed
US-6403792-B1 INHIBIT PRODUCTION OF CASPASE 3 AND 7 IN MAMMALS SMITHKLINE BEECHAM CORPORATION 2002-06-11 US disclosed
WO-2001022966-A1 CASPASES AND APOPTOSIS SMITHKLINE BEECHAM CORPORATION (US) 2001-04-05 WO disclosed