SCHEMBL6539309

SCHEMBL6539309

CC/C(=C\C(=O)O)c1ccc(OCc2ccccc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.61
NR4A1 P22736 1/20 0.60
NR4A2 P43354 1/20 0.60
NR4A3 Q92570 1/20 0.60
PARP10 Q53GL7 1/20 0.57
LTB4R Q15722 1/20 0.57
LTB4R2 Q9NPC1 1/20 0.57
ALDH1A1 P00352 2/20 0.57
HTT P42858 2/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
RAB9A P51151 2/20 0.57
GAA P10253 1/20 0.57
MAPT P10636 1/20 0.57
SRD5A2 P31213 1/20 0.56
HDAC3 O15379 1/20 0.54
HDAC1 Q13547 1/20 0.54
HDAC2 Q92769 1/20 0.54
NCOR2 Q9Y618 1/20 0.54
PLA2G4B P0C869 1/20 0.54
RXRA P19793 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2498876 0.85 MAOB (0.64) MAOBNR4A1NR4A2NR4A3ALDH1A1
SCHEMBL8913237 0.81 NR4A2 (0.66) MAOBNR4A1NR4A2NR4A3PARP10
SCHEMBL102983 0.80 RAB9A (0.83) MAOBNR4A1NR4A2NR4A3PARP10
SCHEMBL2303273 0.79 PDPK1 (0.51) SMN1; SMN2MAPTHDAC3HDAC1HDAC2
SCHEMBL6515252 0.79 PDPK1 (0.51) SMN1; SMN2MAPTHDAC3HDAC1HDAC2
SCHEMBL2303277 0.79 PDPK1 (0.51) SMN1; SMN2MAPTHDAC3HDAC1HDAC2
SCHEMBL7486774 0.79 ESR1 (0.44) NR4A1NR4A2NR4A3ALDH1A1SMN1; SMN2
SCHEMBL434843 0.79 CA1 (0.53) PARP10ALDH1A1HTTSMN1; SMN2HDAC3
SCHEMBL8474022 0.79 CA1 (0.53) PARP10ALDH1A1HTTSMN1; SMN2HDAC3
SCHEMBL8474020 0.79 CA1 (0.53) PARP10ALDH1A1HTTSMN1; SMN2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6812235-B2 2-ACYLAMINO- BETA -ALANINE DERIVATIVES AND A PHARMACEUTICALLY ACCEPTABLE SALT, USEFUL AS FIBRINOGEN RECEPTOR ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-11-02 US disclosed
US-20030018193-A1 Beta-alanine derivatives and their use as receptor anatgonists ASTELLAS PHARMA INC. (JP) 2003-01-23 US disclosed
EP-1255748-A1 BETA-ALANINE DERIVATIVES AND THEIR USE AS RECEPTOR ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-11-13 EP disclosed
WO-2001060813-A1 BETA-ALANINE DERIVATIVES AND THEIR USE AS RECEPTOR ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-08-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030018193-A1 Beta-alanine derivatives and their use as receptor anatgonists ARRB1, ADRB1, GLRB MAOB 300/4885NR4A1 826/4885NR4A2 995/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.