SCHEMBL6545449

SCHEMBL6545449

CC(=O)Cl.CC(=O)NCC1C2CCC1N(Cc1ccccc1)C2

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 7/20 0.46
MTNR1B P49286 3/20 0.46
BRD4 O60885 1/20 0.43
ROCK2 O75116 1/20 0.42
ARHGDIA P52565 1/20 0.42
ROCK1 Q13464 1/20 0.42
MAPT P10636 1/20 0.41
ALDH1A1 P00352 1/20 0.38
ACHE P22303 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6180405 0.98 MTNR1A (0.47) MTNR1AMTNR1BBRD4ROCK2ARHGDIA
Hydrochloric Acid SCHEMBL6708207 0.96 MTNR1A (0.46) MTNR1AMTNR1BBRD4ROCK2ARHGDIA
SCHEMBL5833927 0.79 ROCK2 (0.43) ROCK2ARHGDIAROCK1MAPT
SCHEMBL5833283 0.76 GBA1 (0.46) ROCK2ARHGDIAROCK1MAPT
SCHEMBL6545036 0.76 ROCK2 (0.43) ROCK2ARHGDIAROCK1MAPTALDH1A1
SCHEMBL5832943 0.76 ALPL (0.54) ACHE
SCHEMBL5833530 0.75 MAPK1 (0.44) ALDH1A1
SCHEMBL6707469 0.75 DRD2 (0.47) ROCK2ARHGDIAROCK1MAPT
Hydrochloric Acid SCHEMBL6709626 0.75 ROCK2 (0.43) ROCK2ARHGDIAROCK1MAPTALDH1A1
Hydrochloric Acid SCHEMBL6709625 0.74 DRD2 (0.46) ROCK2ARHGDIAROCK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379502-A1 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS MERCK PATENT GmbH (DE) 2004-01-14 EP disclosed
WO-2002083640-A1 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS MERCK PATENT GMBH (DE) 2002-10-24 WO disclosed