SCHEMBL654591

SCHEMBL654591

COC(=O)C1CNCCN1C(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.42
NR1H2 P55055 1/20 0.42
NR1H3 Q13133 1/20 0.42
PTPN1 P18031 1/20 0.40
HSD17B10 Q99714 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 1/20 0.38
MC4R P32245 1/20 0.37
MC5R P33032 1/20 0.37
LMNA P02545 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ITGB2 P05107 1/20 0.36
ICAM1 P05362 1/20 0.36
ITGAL P20701 1/20 0.36
FKBP1A P62942 1/20 0.35
SCN4A P35499 1/20 0.34
EPHX2 P34913 1/20 0.34
UCHL1 P09936 1/20 0.34
USP30 Q70CQ3 1/20 0.34
USP2 O75604 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1634791 1.00 PARP1 (0.42) PARP1NR1H2NR1H3PTPN1HSD17B10
SCHEMBL6350612 1.00 PARP1 (0.42) PARP1NR1H2NR1H3PTPN1HSD17B10
Ammonia Solution, Strong SCHEMBL22169218 0.99 PARP1 (0.42) PARP1NR1H2NR1H3PTPN1HSD17B10
Hydrochloric Acid SCHEMBL15645732 0.99 PARP1 (0.42) PARP1NR1H2NR1H3PTPN1HSD17B10
SCHEMBL25572934 0.92 HSD17B10 (0.43) PARP1NR1H2NR1H3PTPN1HSD17B10
SCHEMBL18673224 0.91 PARP1 (0.44) PARP1NR1H2NR1H3HSD17B10SMN1; SMN2
SCHEMBL2584375 0.91 PARP1 (0.44) PARP1NR1H2NR1H3HSD17B10SMN1; SMN2
SCHEMBL28442303 0.88 PARP1 (0.38) PARP1NR1H2NR1H3HSD17B10SMN1; SMN2
SCHEMBL7995550 0.88 PARP1 (0.44) PARP1NR1H2NR1H3HSD17B10SMN1; SMN2
SCHEMBL6198122 0.86 TSHR (0.40) ITGB2ICAM1ITGALFKBP1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 402 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026101698-A1 HEPCIDIN MIMETIC COMPOUNDS AND USES THEREOF PROTAGONIST THERAPEUTICS, INC. (US) 2026-05-15 WO disclosed
CN-117659017-B TRPML1/2 modulator compound, pharmaceutical composition, preparation method and application thereof 北京华益健康药物研究中心 2026-05-15 CN disclosed
EP-4161931-B1 NOVEL IMIDAZOPYRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2026-02-18 EP disclosed
US-20250388585-A1 PRMT5 INHIBITORS AND USES THEREOF GILEAD SCIENCES INC (US) 2025-12-25 US disclosed
US-20250282760-A1 OREXIN RECEPTOR AGONISTS MERCK SHARP & DOHME LLC (US) 2025-09-11 US disclosed
US-20250170248-A1 SMARCA DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. 2025-05-29 US disclosed
US-12286434-B2 Pan-tropic entry inhibitors EMORY UNIVERSITY (US) 2025-04-29 US disclosed
EP-4518853-A1 OREXIN RECEPTOR AGONISTS Merck Sharp & Dohme LLC (US) 2025-03-12 EP disclosed
US-12234244-B2 Substituted piperazines as inhibitors of KRAS G12C ARAXES PHARMA LLC (US) 2025-02-25 US disclosed
EP-4405334-B1 SORTILIN INHIBITORS SORTINA PHARMA AB (SE) 2025-02-12 EP disclosed
EP-1448566-A2 CHEMOKINE RECEPTOR ANTAGONISTS AND METHODS OF USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2004-08-25 EP disclosed
WO-2003045942-A2 CHEMOKINE RECEPTOR ANTAGONISTS AND METHODS OF USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2003-06-05 WO disclosed
EP-1268449-A1 SUBSTITUTED PIPERIDINES AS MELANOCORTIN RECEPTOR AGONISTS Merck & Co., Inc. (US) 2003-01-02 EP disclosed
US-6458790-B2 DIETETICS; ANTIDABETIC AGENTS; SEXUAL DISRDERS MERCK & CO., INC. 2002-10-01 US disclosed
CN-1353691-A Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2002-06-12 CN disclosed
CN-1350520-A Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2002-05-22 CN disclosed
US-20020019523-A1 Substituted piperidines as melanocortin receptor agonists MERCK SHARP & DOHME CORP. 2002-02-14 US disclosed
WO-2001070708-A1 SUBSTITUTED PIPERIDINES AS MELANOCORTIN RECEPTOR AGONISTS MERCK & CO., INC. (US) 2001-09-27 WO disclosed
US-4997836-A Inhibitor of platelet activating factor TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US disclosed
EP-0368670-A1 Trisubstituted piperazine compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1990-05-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250388585-A1 PRMT5 INHIBITORS AND USES THEREOF PRMT1, PRMT5, PRMT6 PARP1 176/4885NR1H2 2419/4885NR1H3 2328/4885
US-12234244-B2 Substituted piperazines as inhibitors of KRAS G12C KRAS, NRAS, HRAS PARP1 1612/4885NR1H2 3336/4885NR1H3 3617/4885
US-20250170248-A1 SMARCA DEGRADERS AND USES THEREOF SMARCA1, SMARCA2, SMARCC2 PARP1 101/4885NR1H2 2901/4885NR1H3 2749/4885
US-20250282760-A1 OREXIN RECEPTOR AGONISTS HCRTR2, HCRTR1, OXTR PARP1 4754/4885NR1H2 61/4885NR1H3 79/4885
US-12286434-B2 Pan-tropic entry inhibitors CXCR4, CCR5, CXCL12 PARP1 630/4885NR1H2 297/4885NR1H3 238/4885
US-20020019523-A1 Substituted piperidines as melanocortin receptor agonists MC4R, MC5R, MC3R PARP1 1985/4885NR1H2 2191/4885NR1H3 2250/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.