SCHEMBL655272

SCHEMBL655272

CC(=O)Nc1ccnc(=O)[nH]1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.51
POLB P06746 2/20 0.50
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
MAPT P10636 1/20 0.47
CTDSP1 Q9GZU7 1/20 0.47
KMT2A Q03164 4/20 0.42
PTK2 Q05397 1/20 0.40
GAA P10253 2/20 0.39
TP53 P04637 1/20 0.39
KDM4E B2RXH2 2/20 0.38
MEN1 O00255 1/20 0.38
PRNP P04156 1/20 0.38
S100A4 P26447 1/20 0.38
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1827087 0.98 KCNH2 (0.50) KCNH2POLBNPC1RAB9AMAPT
SCHEMBL2463454 0.82 POLB (0.47) KCNH2POLBNPC1RAB9AMAPT
N4-Hydroxycytosine SCHEMBL31006505 0.76
SCHEMBL4412558 0.75 SMN1; SMN2 (0.46) POLBNPC1RAB9AMAPTKMT2A
SCHEMBL3451050 0.71
SCHEMBL31685701 0.70 GAA (0.48) POLBKMT2AGAAKDM4EMEN1
SCHEMBL13135968 0.69 HSD17B10 (0.42) POLBMAPTGAAKDM4EHSP90AA1
Nitric Acid SCHEMBL16448333 0.69 POLB (0.45) KCNH2POLBNPC1RAB9AMAPT
SCHEMBL1358942 0.68 RXFP1 (0.43) POLBMAPTKMT2APTK2GAA
SCHEMBL3797719 0.67 KDM4E (0.37) POLBMAPTKMT2APTK2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 238 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3980554-A1 HYBRIDIZING ALL-LNA OLIGONUCLEOTIDES F. Hoffmann-La Roche AG (CH) 2022-04-13 EP claimed
CN-119019837-B Self-repairing material assembled by nucleobase pairs and preparation method and application thereof 中国科学院宁波材料技术与工程研究所 2026-05-12 CN disclosed
WO-2025072862-A9 OLIGONUCLEOTIDE COMPOSITIONS AND METHODS THEREOF WAVE LIFE SCIENCES LTD. (SG) 2025-06-26 WO disclosed
WO-2025137486-A1 CAP COMPOUNDS AND RNAS COMPRISING THE SAME HELIX NANOTECHNOLOGIES INC (US) 2025-06-26 WO disclosed
WO-2025072862-A1 OLIGONUCLEOTIDE COMPOSITIONS AND METHODS THEREOF WAVE LIFE SCIENCES LTD. (SG) 2025-04-03 WO disclosed
WO-2025042722-A1 PROMOTER PROXIMAL SEQUENCES AND USES THEREOF FOR RNA MANUFACTURING HELIX NANOTECHNOLOGIES INC (US) 2025-02-27 WO disclosed
US-20240420843-A1 METAEPIGENOMICS-BASED DISEASE DIAGNOSTICS Universal Diagnostics, S.A. (ES) 2024-12-19 US disclosed
CN-119019837-A Self-repairing material assembled by nucleobase pairs and preparation method and application thereof 中国科学院宁波材料技术与工程研究所 2024-11-26 CN disclosed
EP-4413154-A2 METAEPIGENOMICS-BASED DISEASE DIAGNOSTICS Micronoma, Inc. (US) 2024-08-14 EP disclosed
CN-118147100-A N-deoxyribotransferase C1 mutant and application thereof in 2' -deoxyribose transfer 上海合全药物研发有限公司 2024-06-07 CN disclosed
EP-1534286-A1 METHODS OF TREATING OR PREVENTING AUTOIMMUNE DISEASES WITH 2,4-PYRIMIDINEDIAMINE COMPOUNDS Rigel Pharmaceuticals, Inc. (US) 2005-06-01 EP disclosed
US-20050113398-A1 Use of 5-halo or trifluoromethylpyrimidine-2,4-diamine compounds to treat proliferative diseases such as tumorgenic cancers RIGEL PHARMACEUTICALS, INC. 2005-05-26 US disclosed
WO-2005016893-A2 2,4-PYRIMIDINEDIAMINE COMPOUNDS FOR USE IN THE TREATMENT OR PREVENTION OF AUTOIMMUNE DISEASES RIGEL PHARMACEUTICALS, INC. (US) 2005-02-24 WO disclosed
WO-2005013996-A2 2,4-PYRIMIDINEDIAMINE COMPOUNDS AND USES AS ANTI-PROLIFERATIVE AGENTS RIGEL PHARMACEUTICALS, INC. (US) 2005-02-17 WO disclosed
US-20050038243-A1 Prevent immunoglobulin receptors signaling cascading; prevention diseases; drugs; antiinflammatory agents MIDCAP FINANCIAL TRUST 2005-02-17 US disclosed
WO-2005012294-A1 2,4-PYRIMIDINEDIAMINE COMPOUNDS FOR USE IN THE TREATMENT OR PREVENTION OF AUTOIMMUNE DISEASES RIGEL PHARMACEUTICALS, INC. (US) 2005-02-10 WO disclosed
EP-1471915-A2 2,4-PYRIMIDINEDIAMINE COMPOUNDS AND THEIR USES Rigel Pharmaceuticals, Inc. (US) 2004-11-03 EP disclosed
WO-2004014382-A1 METHODS OF TREATING OR PREVENTING AUTOIMMUNE DISEASES WITH 2,4-PYRIMIDINEDIAMINE COMPOUNDS RIGEL PHARMACEUTICALS (US) 2004-02-19 WO disclosed
US-20040029902-A1 Antiinflamamtory agents MIDCAP FINANCIAL TRUST 2004-02-12 US disclosed
WO-2003063794-A2 2,4-PYRIMIDINEDIAMINE COMPOUNDS AND THEIR USES RIGEL PHARMACEUTICALS, INC. (US) 2003-08-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040029902-A1 Antiinflamamtory agents FCER2, FCGR1A, HNMT KCNH2 4735/4885POLB 1652/4885NPC1 4203/4885
US-20050038243-A1 Prevent immunoglobulin receptors signaling cascading; prevention diseases; drugs; antiinflammatory agents FCER2, FCGR1A, FCGR2A KCNH2 4299/4885POLB 4509/4885NPC1 2094/4885
US-20050113398-A1 Use of 5-halo or trifluoromethylpyrimidine-2,4-diamine compounds to treat proliferative diseases such as tumorgenic cancers MKI67, DPYD, VHL KCNH2 3694/4885POLB 175/4885NPC1 2190/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.