SCHEMBL6553983

SCHEMBL6553983

CC(=O)Oc1ccc(S(=O)(=O)c2ccc(C[C@@H](C)NC(=O)C(F)(F)F)cc2)cc1C

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.43
ESR1 P03372 1/20 0.41
KCNH2 Q12809 1/20 0.41
CNR1 P21554 1/20 0.38
ACACB O00763 10/20 0.38
GAA P10253 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
PKM P14618 1/20 0.36
ABCC9 O60706 1/20 0.34
ABCC8 Q09428 1/20 0.34
KCNJ11 Q14654 1/20 0.34
KCNJ8 Q15842 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6553980 0.90 ESR1 (0.40) KMT2AESR1KCNH2CNR1ACACB
SCHEMBL6552876 0.90 ESR1 (0.39) KMT2AESR1KCNH2CNR1ACACB
SCHEMBL6541239 0.90 CNR1 (0.44) ESR1KCNH2CNR1ACACB
SCHEMBL6539921 0.87 ESR1 (0.38) ESR1KCNH2CNR1ACACBGAA
SCHEMBL6541355 0.86 PTPN1 (0.46) ACACB
SCHEMBL6554558 0.85 POLB (0.54) KMT2AESR1KCNH2CNR1ACACB
SCHEMBL6540853 0.84 ESR1 (0.42) ESR1KCNH2CNR1ACACBGAA
SCHEMBL6552531 0.84 ESR1 (0.46) ESR1KCNH2CNR1ACACBPOLB
SCHEMBL6552874 0.82 ESR1 (0.38) ESR1KCNH2CNR1ACACBABCC9
SCHEMBL6540840 0.81 NAMPT (0.45) KMT2ACNR1ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1389185-A2 AMINOALCOHOL DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-02-18 EP disclosed
WO-2002094770-A2 AMINOALCOHOL DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-11-28 WO disclosed