SCHEMBL6552874

SCHEMBL6552874

CC(=O)OOc1ccc(S(=O)(=O)c2ccc(C[C@@H](C)NC(=O)C(F)(F)F)cc2)cc1F

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.38
KCNH2 Q12809 1/20 0.38
CNR1 P21554 2/20 0.37
ACACB O00763 7/20 0.37
NAMPT P43490 8/20 0.36
ABCC9 O60706 1/20 0.33
ABCC8 Q09428 1/20 0.33
KCNJ11 Q14654 1/20 0.33
KCNJ8 Q15842 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6553980 0.90 ESR1 (0.40) ESR1KCNH2CNR1ACACBABCC9
SCHEMBL6552876 0.90 ESR1 (0.39) ESR1KCNH2CNR1ACACBNAMPT
SCHEMBL6540840 0.88 NAMPT (0.45) CNR1ACACBNAMPT
SCHEMBL6554555 0.86 ACACB (0.45) ESR1KCNH2CNR1ACACB
SCHEMBL6541730 0.85 CNR1 (0.38) ESR1KCNH2CNR1ACACBNAMPT
SCHEMBL6552529 0.84 ABCC9 (0.44) ESR1KCNH2CNR1ACACBNAMPT
SCHEMBL6541794 0.84 PTPN1 (0.44) CNR1ACACBNAMPT
SCHEMBL6540415 0.82 CNR1 (0.40) ESR1KCNH2CNR1ACACBABCC9
SCHEMBL6553965 0.82 NAMPT (0.37) NAMPT
SCHEMBL6553983 0.82 KMT2A (0.43) ESR1KCNH2CNR1ACACBABCC9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1389185-A2 AMINOALCOHOL DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-02-18 EP disclosed
WO-2002094770-A2 AMINOALCOHOL DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-11-28 WO disclosed