SCHEMBL6554085

SCHEMBL6554085

O=C(O)N1CCC(S(=O)(=O)Cl)CC1

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SPR P35270 1/20 0.32
ALDH1A1 P00352 2/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
HSD11B1 P28845 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27197937 0.88 SPR (0.31) SPR
SCHEMBL4183478 0.88 SPR (0.31) SPR
SCHEMBL20601948 0.81 EPHX2 (0.42) MEN1KMT2A
SCHEMBL20213981 0.79
SCHEMBL1006759 0.78 TSHR (0.36) SPRALDH1A1
SCHEMBL14157439 0.78 CA12 (0.33) SPR
SCHEMBL2771480 0.75 ADRB3 (0.39) ALDH1A1
SCHEMBL28615553 0.74 HSD11B1 (0.34) HSD11B1
SCHEMBL146591 0.74 MAPT (0.37) ALDH1A1MEN1KMT2A
SCHEMBL4651751 0.74 LMNA (0.33) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024110215-A1 PESTICIDALLY ACTIVE CYCLIC AMINE COMPOUNDS SYNGENTA CROP PROTECTION AG (CH) 2024-05-30 WO disclosed
EP-4323343-A2 PYRIDINE DERIVATIVES AND THEIR USE AS PESTICIDE Syngenta Crop Protection AG (CH) 2024-02-21 EP disclosed
US-20230083376-A1 BRM Targeting Compounds And Associated Methods Of Use PRELUDE THERAPEUTICS, INCORPORATED 2023-03-16 US disclosed
US-11084814-B2 Pyrido[3, 4-d]pyrimidine derivative and pharmaceutically acceptable salt thereof TEIJIN PHARMA LIMITED (JP) 2021-08-10 US disclosed
EP-3813813-A1 COMPOUNDS CTXT Pty Limited (AU) 2021-05-05 EP disclosed
EP-3546458-B1 ((PYRIDIN-2-YL)-AMINO)PYRIDO[3,4-D]PYRIMIDINE AND ((PYRIDAZIN-3-YL)-AMINO)PYRIDO[3,4-D]PYRIMIDINE DERIVATIVES AS CDK4/6 INHIBITORS FOR TREATING E.G. RHEUMATOID ARTHRITIS, ARTERIOSCLEROSIS, PULMONARY FIBROSIS, CEREBRAL INFARCTION OR CANCER TEIJIN PHARMA LTD (JP) 2021-01-06 EP disclosed
CN-111094269-A Heterocyclylmethylene derivatives and their use as mGluR5 receptor modulators 瑞蔻达蒂化学制药公司 2020-05-01 CN disclosed
EP-3546458-A1 PYRIDO[3, 4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF Teijin Pharma Limited (JP) 2019-10-02 EP disclosed
CN-101331115-A Derivatives for modulating ion channels VERTEX PHARMA (US) 2008-12-24 CN disclosed
EP-1487803-A1 INDAZOLES SUBSTITUTED WITH AN ANTI-CANCEROUS ACTIVITY Aventis Pharma S.A. (FR) 2004-12-22 EP disclosed
WO-2003078402-A1 INDAZOLES SUBSTITUTED WITH AN ANTI-CANCEROUS ACTIVITY AVENTIS PHARMA S.A. (FR) 2003-09-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230083376-A1 BRM Targeting Compounds And Associated Methods Of Use ADRM1, BRDT, RBX1 SPR 1360/4885ALDH1A1 4038/4885MEN1 3067/4885
US-11084814-B2 Pyrido[3, 4-d]pyrimidine derivative and pharmaceutically acceptable salt thereof CDK4, CDK6, CDK16 SPR 2952/4885ALDH1A1 964/4885MEN1 2438/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.