SCHEMBL6555534

SCHEMBL6555534

O=c1[nH]c2cc(CCN3CCN(c4ccc(Cl)cc4)CC3)ccc2c2c1CCCC2

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.54
PARP1 P09874 14/20 0.53
TNK1 Q13470 10/20 0.52
TNK2 Q07912 6/20 0.52
KCNH2 Q12809 1/20 0.52
PARP2 Q9UGN5 1/20 0.52
ADRA1D P25100 1/20 0.48
ADRA1A P35348 1/20 0.48
ADRA1B P35368 1/20 0.48
HTR1A P08908 3/20 0.46
HTR2A P28223 2/20 0.46
HTR2C P28335 1/20 0.45
DRD1 P21728 1/20 0.45
DRD5 P21918 1/20 0.45
DRD3 P35462 1/20 0.45
TMEM97 Q5BJF2 1/20 0.45
SIGMAR1 Q99720 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6411449 0.99 DRD2 (0.53) DRD2PARP1TNK1TNK2KCNH2
SCHEMBL6405680 0.89 PARP1 (0.64) PARP1TNK1TNK2KCNH2PARP2
SCHEMBL6403556 0.81 PARP1 (0.49) PARP1TNK1TNK2KCNH2PARP2
Hydrochloric Acid SCHEMBL6403678 0.80 PARP1 (0.55) PARP1KCNH2PARP2HTR1ASIGMAR1
Hydrochloric Acid SCHEMBL6403655 0.76 PARP1 (0.60) PARP1KCNH2PARP2SIGMAR1
Hydrochloric Acid SCHEMBL6406350 0.74 PARP1 (0.79) PARP1TNK1TNK2KCNH2PARP2
SCHEMBL6407854 0.74 PARP1 (0.51) PARP1TNK1TNK2KCNH2PARP2
SCHEMBL6556204 0.73 PARP1 (0.53) PARP1TNK1TNK2KCNH2PARP2
SCHEMBL6406366 0.72 PARP1 (0.62) DRD2PARP1TNK1TNK2KCNH2
SCHEMBL25822114 0.72 PARP1 (0.74) PARP1TNK1TNK2KCNH2PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487800-A1 PHENANTHRIDINONES AS PARP INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-12-22 EP disclosed
WO-2003080581-A1 PHENANTHRIDINONES AS PARP INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-10-02 WO disclosed