SCHEMBL6556372

SCHEMBL6556372

CCOC(Cn1c(-c2cc([N+](=O)[O-])cc([N+](=O)[O-])c2)ncc(C(=O)O)c1=O)OCC

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.36
FOS P01100 1/20 0.36
JUN P05412 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
ATM Q13315 1/20 0.35
TP53 P04637 1/20 0.34
HTT P42858 1/20 0.34
ALDH1A1 P00352 3/20 0.34
RAB9A P51151 2/20 0.34
MAPT P10636 2/20 0.34
NPC1 O15118 1/20 0.34
NPBWR1 P48145 1/20 0.34
MCHR1 Q99705 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
LMNA P02545 2/20 0.34
POLB P06746 3/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6556267 0.91 FOS (0.43) FOSJUNNFKB1NFKB2RELA
SCHEMBL6558245 0.90 MAPT (0.40) HTTALDH1A1RAB9AMAPTNPC1
SCHEMBL6556361 0.82 MAPT (0.42) NFKB1NFKB2RELAATMTP53
SCHEMBL6556255 0.81 MAPT (0.46) HTTALDH1A1RAB9AMAPTSMN1; SMN2
SCHEMBL6556282 0.81 KDM4E (0.38) ALDH1A1RAB9AMAPTNPC1SMN1; SMN2
SCHEMBL6557546 0.80 CTRC (0.42) ALDH1A1MAPTMEN1KMT2AGLA
SCHEMBL6556504 0.80 CSNK1D (0.37) FOSJUNNFKB1NFKB2RELA
SCHEMBL6557511 0.79 P2RX3 (0.41) FOSJUNNFKB1NFKB2RELA
SCHEMBL6556234 0.79 ELANE (0.39) FOSJUNNFKB1NFKB2RELA
SCHEMBL6558138 0.78 KDM4E (0.50) FOSJUNNFKB1NFKB2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0826671-B1 HETEROCYCLIC AMIDE COMPOUNDS AND MEDICINAL USE OF THE SAME MITSUBISHI PHARMA CORP (JP) 2004-12-29 EP disclosed
US-5948785-A USEFUL AS CHYMASE INHIBITORS AND CAN BE EFFECTIVE FOR THE PROPHYLAXIS AND TREATMENT OF VARIOUS DISEASES CAUSED BY CHYMASE, SUCH AS THOSE CAUSED BY ANGIOTENSIN II. THE GREEN CROSS CORPORATION (JP) 1999-09-07 US disclosed
EP-0826671-A1 HETEROCYCLIC AMIDE COMPOUNDS AND MEDICINAL USE OF THE SAME THE GREEN CROSS CORPORATION (JP) 1998-03-04 EP disclosed