SCHEMBL6557100

SCHEMBL6557100

CCCOc1cc(C=O)cc(OCCC)c1I

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FDPS P14324 1/20 0.46
ALDH1A1 P00352 10/20 0.41
KDM4E B2RXH2 3/20 0.40
MAPT P10636 5/20 0.38
NPSR1 Q6W5P4 2/20 0.38
HTT P42858 2/20 0.38
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 4/20 0.38
HPGD P15428 4/20 0.38
TDP1 Q9NUW8 3/20 0.38
TP53 P04637 2/20 0.37
GAA P10253 2/20 0.36
TUBB4A P04350 1/20 0.36
TUBB P07437 1/20 0.36
TUBA3C P0DPH7 1/20 0.36
TUBA1B P68363 1/20 0.36
TUBA4A P68366 1/20 0.36
TUBB4B P68371 1/20 0.36
TUBB3 Q13509 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1121574 0.85 ALDH1A1 (0.56) FDPSALDH1A1KDM4EMAPTNPSR1
SCHEMBL16056145 0.85 FDPS (0.38) FDPSALDH1A1KDM4EMAPTNPSR1
SCHEMBL9097669 0.83 FDPS (0.47) FDPSALDH1A1KDM4EMAPTNPSR1
SCHEMBL4217049 0.82 FDPS (0.56) FDPSALDH1A1KDM4EMAPTNPSR1
SCHEMBL5882634 0.78 FDPS (0.69) FDPSALDH1A1KDM4EMAPTNPSR1
SCHEMBL7844422 0.77 TUBB1 (0.57) FDPSALDH1A1KDM4EMAPTNPSR1
SCHEMBL8110374 0.77 ALDH1A1 (0.47) FDPSALDH1A1KDM4EMAPTNPSR1
SCHEMBL7466433 0.76 FDPS (0.53) FDPSALDH1A1KDM4EMAPTNPSR1
SCHEMBL9065484 0.76 KDM4E (0.48) FDPSALDH1A1KDM4EL3MBTL1HPGD
SCHEMBL15567583 0.76 ALOX5 (0.55) FDPSALDH1A1KDM4EMAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230224-B1 SUBSTITUTED 5-BENZYL-2,4-DIAMINOPYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2004-12-29 EP disclosed
US-6821980-B1 Substituted 5-benzyl-2,4-diaminopyrimidines BASILEA PHARMACEUTICA AG (CH) 2004-11-23 US disclosed
EP-1230224-A1 SUBSTITUTED 5-BENZYL-2,4-DIAMINOPYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 2002-08-14 EP disclosed
WO-2001032633-A1 SUBSTITUTED 5-BENZYL-2,4-DIAMINOPYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2001-05-10 WO disclosed