SCHEMBL6558265

SCHEMBL6558265

Brc1cccc(C2OCCO2)c1.COc1ccc(Sc2cccc(C=O)c2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
HTR2C P28335 1/20 0.36
XDH P47989 2/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PTGIR P43119 1/20 0.34
ATM Q13315 1/20 0.34
CYP2A6 P11509 1/20 0.33
EGFR P00533 1/20 0.33
MGLL Q99685 2/20 0.33
KDM4E B2RXH2 1/20 0.32
POLB P06746 1/20 0.31
APP P05067 1/20 0.31
MEN1 O00255 1/20 0.31
USP2 O75604 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6558248 0.88 ALDH1A1 (0.44) ALDH1A1TDP1MAOAMAOBCYP2A6
SCHEMBL6557103 0.83 ALDH1A1 (0.37) ALDH1A1RAB9ASMN1; SMN2KDM4EAPP
SCHEMBL6557408 0.82 ALDH1A1 (0.45) ALDH1A1NPC1RAB9AMAOAMAOB
SCHEMBL6255853 0.80 NPC1 (0.52) ALDH1A1NPC1RAB9ATDP1HTR2C
SCHEMBL2281435 0.71 ALDH1A1 (0.42) ALDH1A1TDP1MAOAMAOBSMN1; SMN2
SCHEMBL4800339 0.70 NPC1 (0.50) ALDH1A1NPC1RAB9ATDP1CYP2A6
SCHEMBL194639 0.70 KDM1A (0.50) ALDH1A1HTR2CPOLBMEN1KMT2A
SCHEMBL6159034 0.69 SRC (0.42) ALDH1A1NPC1RAB9ATDP1MAOA
SCHEMBL2532959 0.68 SLC5A2 (0.50) NPC1RAB9ATDP1HTR2CATM
SCHEMBL1680858 0.68 MEN1 (0.40) NPC1RAB9AHTR2CMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392643-A2 TRISUBSTITUTED-N- (1S)-1,2,3,4-TETRAHYDRO-1-NAPHTHALENYL] BENZAMIDES WHICH INHIBIT P2X3 AND P2X2/3 CONTAINING RECEPTORS Abbott Laboratories (US) 2004-03-03 EP disclosed
WO-2002094767-A2 TRISUBSTITUTED-N-[(1S)-1,2,3,4-TETRAHYDRO-1-NAPHTHALENYL] BENZAMIDES WHICH INHIBIT P2X3 AND P2X2/3 CONTAINING RECEPTORS ABBOTT LABORATORIES (US) 2002-11-28 WO disclosed