SCHEMBL6557408

SCHEMBL6557408

Brc1cccc(C2OCCO2)c1.CSc1cccc(C=O)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
ATM Q13315 1/20 0.38
MAOA P21397 2/20 0.34
MAOB P27338 2/20 0.34
MAPK1 P28482 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
KDM1A O60341 4/20 0.33
RCOR1 Q9UKL0 2/20 0.33
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
TUBA1B P68363 1/20 0.33
TUBA4A P68366 1/20 0.33
TUBB4B P68371 1/20 0.33
TUBB3 Q13509 1/20 0.33
TUBB2A Q13885 1/20 0.33
TUBB8 Q3ZCM7 1/20 0.33
TUBA3E Q6PEY2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6558248 0.87 ALDH1A1 (0.44) ALDH1A1MAOAMAOBKDM1ARCOR1
SCHEMBL6558265 0.82 ALDH1A1 (0.38) ALDH1A1NPC1RAB9AATMMAOA
SCHEMBL6557103 0.80 ALDH1A1 (0.37) ALDH1A1RAB9AMAPK1SMN1; SMN2MEN1
SCHEMBL17860605 0.78 RAB9A (0.45) ALDH1A1NPC1RAB9AATMMAPK1
SCHEMBL2281435 0.78 ALDH1A1 (0.42) ALDH1A1MAOAMAOBSMN1; SMN2DRD2
SCHEMBL194639 0.77 KDM1A (0.50) ALDH1A1MAPK1KDM1ARCOR1DRD2
SCHEMBL29951214 0.75 ALDH1A1 (0.56) ALDH1A1NPC1RAB9AMAPK1TUBB4A
SCHEMBL711416 0.75 ALDH1A1 (0.56) ALDH1A1NPC1RAB9AMAPK1TUBB4A
SCHEMBL29995306 0.72 DRD2 (0.42) ALDH1A1NPC1RAB9AATMMAOA
SCHEMBL6196036 0.72 DRD2 (0.42) ALDH1A1NPC1RAB9AATMMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392643-A2 TRISUBSTITUTED-N- (1S)-1,2,3,4-TETRAHYDRO-1-NAPHTHALENYL] BENZAMIDES WHICH INHIBIT P2X3 AND P2X2/3 CONTAINING RECEPTORS Abbott Laboratories (US) 2004-03-03 EP disclosed
WO-2002094767-A2 TRISUBSTITUTED-N-[(1S)-1,2,3,4-TETRAHYDRO-1-NAPHTHALENYL] BENZAMIDES WHICH INHIBIT P2X3 AND P2X2/3 CONTAINING RECEPTORS ABBOTT LABORATORIES (US) 2002-11-28 WO disclosed