SCHEMBL6558475

SCHEMBL6558475

CC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@@H](CC(=O)N(C)C)C(=O)NC(C)C(=O)C(F)(F)F)C(C)(C)C(=O)O)C(C)C

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PSENEN Q9NZ42 1/20 0.32
CASP3 P42574 1/20 0.32
CASP2 P42575 1/20 0.32
CASP1 P29466 1/20 0.31
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6558459 0.92 ADAM17 (0.35) PSENENCASP1BACE1
SCHEMBL6558839 0.89 PSENEN (0.36) PSENENCASP3CASP2CASP1BACE1
SCHEMBL6558973 0.86 PSENEN (0.36) PSENENCASP3CASP2CASP1BACE1
SCHEMBL6558456 0.86 PSENEN (0.37) PSENENCASP1BACE1
SCHEMBL6558461 0.84 RRM1 (0.33)
SCHEMBL6558875 0.79 CASP1 (0.42) PSENENCASP3CASP2CASP1BACE1
SCHEMBL6558467 0.77 MEN1 (0.31) CASP3
SCHEMBL8001329 0.77 CAPN1 (0.35) CASP1
SCHEMBL6558829 0.76 MMP1 (0.32)
SCHEMBL6558489 0.76 CASP1 (0.36) CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948523-B1 PEPTIDOMIMETIC INHIBITORS OF THE HUMAN CYTOMEGALOVIRUS PROTEASE BOEHRINGER INGELHEIM CA LTD (CA) 2004-03-17 EP claimed
US-6291640-B1 OLIGOPEPTIDES; SOLID PHASE SYNTHESIS BOEHRINGER INGELHEIM LTD. (CA) 2001-09-18 US claimed
EP-0948523-B1 PEPTIDOMIMETIC INHIBITORS OF THE HUMAN CYTOMEGALOVIRUS PROTEASE BOEHRINGER INGELHEIM CA LTD (CA) 2004-03-17 EP disclosed
US-6291640-B1 OLIGOPEPTIDES; SOLID PHASE SYNTHESIS BOEHRINGER INGELHEIM LTD. (CA) 2001-09-18 US disclosed