SCHEMBL6558478

SCHEMBL6558478

CC(C)C[C@H](NC(=O)[C@@H](N)CCCN)C(=O)N[C@@H](CO)[C@@H](O)[C@@H](O)[C@H](O)C(=O)N[C@@H](CC(=O)O)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 2/20 0.42
METAP1 P53582 2/20 0.42
BACE1 P56817 11/20 0.41
BACE2 Q9Y5Z0 3/20 0.41
OPRK1 P41145 1/20 0.38
ERAP2 Q6P179 2/20 0.37
CTSD P07339 2/20 0.37
IL1RN P18510 1/20 0.37
REN P00797 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6559233 0.97 METAP2 (0.41) METAP2METAP1BACE1BACE2OPRK1
Hydrochloric Acid SCHEMBL6559317 0.92 REN (0.43) METAP2METAP1BACE1BACE2ERAP2
SCHEMBL6558490 0.91 BACE1 (0.49) METAP2METAP1BACE1BACE2ERAP2
SCHEMBL6560842 0.91 METAP2 (0.43) METAP2METAP1BACE1BACE2ERAP2
SCHEMBL6559229 0.91 METAP2 (0.45) METAP2METAP1BACE1BACE2ERAP2
Hydrochloric Acid SCHEMBL6560796 0.91 METAP2 (0.43) METAP2METAP1BACE1BACE2ERAP2
Hydrochloric Acid SCHEMBL6559352 0.90 METAP2 (0.44) METAP2METAP1
Hydrochloric Acid SCHEMBL6559362 0.90 METAP2 (0.44) METAP2METAP1
SCHEMBL6559296 0.90 BACE1 (0.44) METAP2METAP1BACE1BACE2CTSD
SCHEMBL6559264 0.89 METAP2 (0.42) METAP2METAP1BACE1BACE2ERAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998488-B1 POLYOL-AMINO ACID COMPOUNDS HAVING ANTI-HELICOBACTER PYLORI ACTIVITY TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2004-03-17 EP disclosed
US-6423869-B1 BACTERICIDES, ANTIULCER AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-07-23 US disclosed