SCHEMBL6558490

SCHEMBL6558490

CC(C)C[C@H](NC(=O)[C@@H](N)CCC(=O)O)C(=O)N[C@@H](CO)[C@@H](O)[C@@H](O)[C@H](O)C(=O)N[C@@H](CC(=O)O)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 16/20 0.49
BACE2 Q9Y5Z0 5/20 0.49
METAP2 P50579 2/20 0.43
METAP1 P53582 2/20 0.43
ERAP2 Q6P179 1/20 0.43
CTSD P07339 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6559296 0.95 BACE1 (0.44) BACE1BACE2METAP2METAP1CTSD
SCHEMBL6559229 0.93 METAP2 (0.45) BACE1BACE2METAP2METAP1ERAP2
Hydrochloric Acid SCHEMBL6560796 0.92 METAP2 (0.43) BACE1BACE2METAP2METAP1ERAP2
SCHEMBL6558478 0.91 METAP2 (0.42) BACE1BACE2METAP2METAP1ERAP2
SCHEMBL6560842 0.91 METAP2 (0.43) BACE1BACE2METAP2METAP1ERAP2
Hydrochloric Acid SCHEMBL6559317 0.91 REN (0.43) BACE1BACE2METAP2METAP1ERAP2
SCHEMBL6559264 0.91 METAP2 (0.42) BACE1BACE2METAP2METAP1ERAP2
SCHEMBL6558505 0.91 METAP2 (0.46) BACE1BACE2METAP2METAP1ERAP2
SCHEMBL6558918 0.90 METAP2 (0.47) BACE1BACE2METAP2METAP1ERAP2
Hydrochloric Acid SCHEMBL6558938 0.90 METAP2 (0.43) BACE1BACE2METAP2METAP1ERAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998488-B1 POLYOL-AMINO ACID COMPOUNDS HAVING ANTI-HELICOBACTER PYLORI ACTIVITY TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2004-03-17 EP disclosed
US-6423869-B1 BACTERICIDES, ANTIULCER AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-07-23 US disclosed