SCHEMBL6559028

SCHEMBL6559028

COc1ccc2nccc(CCCNC(C)=O)c2c1

nearest known ligand 0.86

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 16/20 0.86
MTNR1A P48039 15/20 0.86
HTR2C P28335 1/20 0.54
HTR2B P41595 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6559881 0.93 MTNR1B (1.00) MTNR1BMTNR1AHTR2CHTR2B
SCHEMBL6560437 0.82 MTNR1A (0.60) MTNR1BMTNR1AHTR2CHTR2B
SCHEMBL6559038 0.81 MTNR1A (1.00) MTNR1BMTNR1A
SCHEMBL20542004 0.81 MTNR1A (0.63) MTNR1BMTNR1A
SCHEMBL6558990 0.79 MTNR1A (0.75) MTNR1BMTNR1A
SCHEMBL592246 0.79 MTNR1A (0.67) MTNR1BMTNR1A
SCHEMBL30449211 0.78 MTNR1A (0.73) MTNR1BMTNR1AHTR2CHTR2B
SCHEMBL29032157 0.78 MTNR1A (0.73) MTNR1BMTNR1AHTR2CHTR2B
SCHEMBL6560401 0.78 MTNR1A (0.74) MTNR1BMTNR1A
SCHEMBL8031017 0.78 MTNR1A (0.86) MTNR1BMTNR1AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0837850-B1 4-ACYLAMINO(HALOGENO) ALKYL-QUINOLINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MELATONIN AGONISTS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2004-09-01 EP disclosed
EP-0837850-A1 4-ACYLAMINO(HALOGENO) ALKYL-QUINOLINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MELATONIN AGONISTS Takeda Chemical Industries, Ltd. (JP) 1998-04-29 EP disclosed
US-5708005-A MELATONIN RECEPTOR BINDERS, SLEEP DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-01-13 US disclosed
WO-1997001539-A1 4-ACYLAMINO(HALOGENO) ALKYL-QUINOLINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MELATONIN AGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-01-16 WO disclosed