SCHEMBL6560042

SCHEMBL6560042

CS/C(=N\C(C)=O)NC(C)=O

nearest known ligand 0.35

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 1/20 0.35
TAS2R38 P59533 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10170621 1.00 CRBN (0.35) CRBNTAS2R38
SCHEMBL6560044 1.00 CRBN (0.35) CRBNTAS2R38
SCHEMBL11698336 0.84 CRBN (0.33) CRBNTAS2R38
SCHEMBL25480034 0.80 SMN1; SMN2 (0.31)
SCHEMBL3753647 0.78
SCHEMBL13219908 0.78
SCHEMBL3753641 0.78
SCHEMBL15084705 0.77
SCHEMBL10329427 0.76 ALDH1A1 (0.31)
SCHEMBL21359614 0.74 DGAT1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023239007-A1 BENZIMIDAZOLE DERIVATIVE, PREPARATION METHOD THEREOF, AND PHARMACEUTICAL COMPOSITION FOR PREVENTION OR TREATMENT OF CANCER OR INFECTIOUS DISEASES CONTAINING SAME AS ACTIVE INGREDIENT 한국화학연구원 2023-12-14 WO disclosed
WO-2023239007-A1 BENZIMIDAZOLE DERIVATIVE, PREPARATION METHOD THEREOF, AND PHARMACEUTICAL COMPOSITION FOR PREVENTION OR TREATMENT OF CANCER OR INFECTIOUS DISEASES CONTAINING SAME AS ACTIVE INGREDIENT 한국화학연구원 2023-12-14 WO disclosed
US-11708352-B2 Anti-cancer compounds THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-07-25 US disclosed
US-20220267307-A1 ANTI-CANCER COMPOUNDS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2022-08-25 US disclosed
US-10562886-B2 Anti-cancer compounds THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2020-02-18 US disclosed
US-20180354932-A1 ANTI-CANCER COMPOUNDS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2018-12-13 US disclosed
US-9937192-B2 Combination therapy to treat mycobacterium diseases SPERO TRINEM, INC. (US) 2018-04-10 US disclosed
US-20170128471-A1 COMBINATION THERAPY TO TREAT MYCOBACTERIUM DISEASES SPERO THERAPEUTICS, INC. 2017-05-11 US disclosed
US-20160289175-A1 CREATINE ANALOGS AND THE USE THEREOF ULTRAGENYX PHARMACEUTICAL INC. 2016-10-06 US disclosed
EP-1391454-B1 Substituted benzamide compounds with antihypertensive activity MITSUBISHI TANABE PHARMA CORP (JP) 2012-05-30 EP disclosed
US-20070249600-A1 CHEMICAL COMPOUNDS CHEUNG MUI 2007-10-25 US disclosed
US-7238813-B2 Chemical compounds SMITHKLINE BEECHAM CORPORATION (US) 2007-07-03 US disclosed
EP-1391454-A1 Substituted benzamide compounds with antihypertensive activity Mitsubishi Pharma Corporation (JP) 2004-02-25 EP disclosed
EP-1195372-A1 N-heterocyclic substituted benzamide derivatives with antihypertensive activity Mitsubishi Pharma Corporation (JP) 2002-04-10 EP disclosed
US-6156766-A Benzamide compounds and pharmaceutical use thereof YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 2000-12-05 US disclosed
EP-0641781-B1 4-AMINO(ALKYL)CYCLOHEXANE-1-CARBOXAMIDE COMPOUND AND USE THEREOF YOSHITOMI PHARMACEUTICAL (JP) 2000-07-26 EP disclosed
US-5958944-A TREATMENT OF CIRCULATORY DISEASES IN CORONARY, CEREBRAL, RENAL AND PERIPHERAL ARTERIES, AS A THERAPEUTIC AGENT FOR HYPERTENSION, ANGINA PECTORIS, AND RENAL AND PERIPHERAL CIRCULATION DISORDER, ANTIASTHMATIC AGENT YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1999-09-28 US disclosed
EP-0757038-A1 BENZAMIDE COMPOUND AND MEDICINAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-02-05 EP disclosed
US-5478838-A Treating hypertension, angina pectoris, asthma, improving peripheral circulation YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1995-12-26 US disclosed
EP-0641781-A1 4-AMINO(ALKYL)CYCLOHEXANE-1-CARBOXAMIDE COMPOUND AND USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1995-03-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10562886-B2 Anti-cancer compounds TP53, VHL, BAD CRBN 1412/4885TAS2R38 4715/4885
US-20070249600-A1 CHEMICAL COMPOUNDS TIE1, KDR, FLT4 CRBN 408/4885TAS2R38 2546/4885
US-20180354932-A1 ANTI-CANCER COMPOUNDS TP53, VHL, BAD CRBN 1412/4885TAS2R38 4715/4885
US-20170128471-A1 COMBINATION THERAPY TO TREAT MYCOBACTERIUM DISEASES TOP1, TOP2A, TOP2B CRBN 4816/4885TAS2R38 4689/4885
US-11708352-B2 Anti-cancer compounds TP53, VHL, BAD CRBN 1412/4885TAS2R38 4715/4885
US-20220267307-A1 ANTI-CANCER COMPOUNDS TP53, VHL, BAD CRBN 1412/4885TAS2R38 4715/4885
US-20160289175-A1 CREATINE ANALOGS AND THE USE THEREOF CKMT1A; CKMT1B, CPT1B, GLS CRBN 1682/4885TAS2R38 3597/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.