SCHEMBL6561597

SCHEMBL6561597

CCCc1c(O)ccc2c(C(C)(C)C)cc(=O)oc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.51
KDM4E B2RXH2 8/20 0.51
HPGD P15428 7/20 0.51
GAA P10253 6/20 0.51
GLA P06280 5/20 0.51
HIF1A Q16665 2/20 0.51
KMT2A Q03164 5/20 0.50
ERAP1 Q9NZ08 5/20 0.50
CASP1 P29466 4/20 0.50
CASP7 P55210 4/20 0.50
MEN1 O00255 3/20 0.50
HSD17B10 Q99714 3/20 0.50
POLB P06746 1/20 0.50
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C19 P33261 1/20 0.49
CSNK2A2 P19784 1/20 0.46
CSNK2B P67870 1/20 0.46
CSNK2A1 P68400 1/20 0.46
USP2 O75604 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1594333 0.88 CSNK2A2 (0.61) ALDH1A1KDM4EHPGDGAAGLA
SCHEMBL11079352 0.82 GAA (0.63) ALDH1A1KDM4EHPGDGAAGLA
SCHEMBL6560136 0.82 KDM4E (0.64) ALDH1A1KDM4EHPGDGAAGLA
SCHEMBL6559997 0.82 GAA (0.71) ALDH1A1KDM4EHPGDGAAGLA
SCHEMBL6561714 0.82 KDM4E (0.58) ALDH1A1KDM4EHPGDGAAGLA
SCHEMBL6559297 0.79 ALDH1A1 (0.34) ALDH1A1KDM4EHPGDGAAGLA
SCHEMBL15211319 0.78 MCL1 (0.66) ALDH1A1KDM4EHPGDGAAGLA
SCHEMBL6561528 0.75 KDM4E (0.49) ALDH1A1KDM4EPOLBMAOB
SCHEMBL14756049 0.75 GAA (0.70) ALDH1A1KDM4EHPGDGAAGLA
SCHEMBL6561715 0.75 ESR2 (0.50) ALDH1A1KDM4EHPGDGAAGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0904079-B1 ANTIDIABETIC AGENTS MERCK & CO INC (US) 2004-03-24 EP disclosed
EP-0904079-A4 1999-05-06 EP disclosed
EP-0904079-A1 ANTIDIABETIC AGENTS Merck & Co., Inc. (US) 1999-03-31 EP disclosed
US-5859051-A ACETYLPHENOL DERIVATIVES MERCK & CO., INC. (US) 1999-01-12 US disclosed
WO-1997027857-A1 ANTIDIABETIC AGENTS MERCK & CO., INC. (US) 1997-08-07 WO disclosed