SCHEMBL6560178

SCHEMBL6560178

CC(C)=COc1ccc2c(-c3ccccc3)coc2c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.66
ALDH1A1 P00352 10/20 0.55
MAPT P10636 7/20 0.55
SMN1; SMN2 Q16637 7/20 0.55
NPC1 O15118 6/20 0.55
RAB9A P51151 5/20 0.55
KDM4E B2RXH2 5/20 0.55
MEN1 O00255 5/20 0.53
KMT2A Q03164 5/20 0.53
HPGD P15428 5/20 0.53
TP53 P04637 4/20 0.53
CYP3A4 P08684 3/20 0.53
POLB P06746 3/20 0.52
MAPK1 P28482 2/20 0.50
GAA P10253 2/20 0.50
HDAC6 Q9UBN7 2/20 0.50
PTGS1 P23219 1/20 0.50
SLC6A2 P23975 1/20 0.50
STAT1 P42224 1/20 0.50
CASP3 P42574 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1742372 0.80 PIN1 (1.00) PIN1ALDH1A1MAPTSMN1; SMN2NPC1
SCHEMBL11421623 0.73 ALDH1A1 (0.69) PIN1ALDH1A1MAPTSMN1; SMN2NPC1
SCHEMBL4884228 0.71 ALDH1A1 (0.77) PIN1ALDH1A1MAPTSMN1; SMN2NPC1
SCHEMBL11546488 0.71 PIN1 (0.64) PIN1ALDH1A1MAPTSMN1; SMN2NPC1
SCHEMBL4887390 0.71 PIN1 (0.63) PIN1ALDH1A1MAPTSMN1; SMN2NPC1
SCHEMBL2070406 0.71 NPC1 (1.00) ALDH1A1MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL5990085 0.70 PIN1 (0.57) PIN1ALDH1A1MAPTSMN1; SMN2NPC1
SCHEMBL10014193 0.70 PIN1 (0.61) PIN1ALDH1A1MAPTSMN1; SMN2NPC1
SCHEMBL762092 0.69 MAPT (1.00) PIN1ALDH1A1MAPTSMN1; SMN2NPC1
SCHEMBL4896442 0.69 ALDH2 (0.64) PIN1ALDH1A1MAPTALDH2MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0904079-B1 ANTIDIABETIC AGENTS MERCK & CO INC (US) 2004-03-24 EP disclosed
EP-0904079-A4 1999-05-06 EP disclosed
EP-0904079-A1 ANTIDIABETIC AGENTS Merck & Co., Inc. (US) 1999-03-31 EP disclosed
US-5859051-A ACETYLPHENOL DERIVATIVES MERCK & CO., INC. (US) 1999-01-12 US disclosed
WO-1997027857-A1 ANTIDIABETIC AGENTS MERCK & CO., INC. (US) 1997-08-07 WO disclosed