SCHEMBL6560700

SCHEMBL6560700

CNC(=O)C=C(Cc1ccc(OC)cc1)c1ccccc1C

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.51
RAB9A P51151 3/20 0.51
TDP1 Q9NUW8 3/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
ATM Q13315 1/20 0.49
LMNA P02545 1/20 0.48
USP2 O75604 1/20 0.48
TP53 P04637 1/20 0.48
ALDH1A1 P00352 4/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
MAPT P10636 1/20 0.45
KDM4E B2RXH2 2/20 0.45
POLB P06746 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
HTT P42858 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
KLK7 P49862 2/20 0.44
FFAR1 O14842 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6560672 0.84 CACNA1B (0.52) NPC1RAB9ATDP1L3MBTL1USP2
SCHEMBL6561877 0.78 NPC1 (0.51) NPC1RAB9AL3MBTL1LMNAALDH1A1
SCHEMBL6560697 0.78 NPC1 (0.51) NPC1RAB9AL3MBTL1LMNAALDH1A1
SCHEMBL6561872 0.75 ALDH1A1 (0.52) NPC1RAB9ATDP1LMNATP53
SCHEMBL4569297 0.70 HPGD (0.69) NPC1RAB9ALMNATP53ALDH1A1
SCHEMBL580634 0.70 USP2 (0.71) NPC1RAB9ATDP1ATMUSP2
SCHEMBL6357074 0.69 KMT2A (0.68) NPC1RAB9ALMNATP53ALDH1A1
SCHEMBL3369060 0.68 HTT (0.76) NPC1RAB9ATDP1LMNAALDH1A1
SCHEMBL10062017 0.68 NPC1 (1.00) NPC1RAB9ALMNAALDH1A1SMN1; SMN2
SCHEMBL7805240 0.67 HTT (0.48) NPC1RAB9ATDP1L3MBTL1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944581-A4 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES LILLY CO ELI (US) 2004-09-08 EP disclosed
EP-0944581-A1 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES ELI LILLY AND COMPANY (US) 1999-09-29 EP disclosed
WO-1998022429-A1 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES ELI LILLY AND COMPANY (US) 1998-05-28 WO disclosed