SCHEMBL6560707

SCHEMBL6560707

C#CC(=O)N(C)c1cc2ccccc2c2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
HPGD P15428 3/20 0.39
MAPT P10636 2/20 0.39
TRPM4 Q8TD43 1/20 0.39
SIGMAR1 Q99720 3/20 0.38
HSD17B10 Q99714 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
CYP1A2 P05177 1/20 0.37
GLA P06280 1/20 0.37
CYP2C19 P33261 1/20 0.37
KMT2A Q03164 1/20 0.37
POLB P06746 1/20 0.37
PKM P14618 1/20 0.37
RAD52 P43351 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
GPR84 Q9NQS5 1/20 0.35
HIF1A Q16665 1/20 0.34
CYP1B1 Q16678 1/20 0.34
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6561817 0.80 SIGMAR1 (0.61) SIGMAR1GAA
SCHEMBL20384970 0.74 TRPM4 (0.33) MAPTTRPM4SIGMAR1POLBPKM
SCHEMBL20384989 0.73 TRPM4 (0.36) MAPTTRPM4SIGMAR1POLBPKM
SCHEMBL3281012 0.73 CHEK1 (0.47) ALDH1A1HPGDMAPTTRPM4SIGMAR1
SCHEMBL6563222 0.70 SIGMAR1 (0.45) ALDH1A1SIGMAR1
SCHEMBL9888945 0.68 ALDH1A1 (0.50) ALDH1A1HPGDMAPTTRPM4HSD17B10
SCHEMBL28476383 0.67 POLB (0.52) KDM4EMEN1KMT2APOLBPKM
SCHEMBL12048720 0.67 TRPM4 (0.41) ALDH1A1HPGDMAPTTRPM4SIGMAR1
SCHEMBL20384969 0.66 TRPM4 (0.34) ALDH1A1TRPM4SIGMAR1HSD17B10GPR84
SCHEMBL12258286 0.66 SIGMAR1 (0.50) ALDH1A1HPGDTRPM4SIGMAR1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944581-A4 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES LILLY CO ELI (US) 2004-09-08 EP disclosed
US-6069247-A REACTING AN ACETYLENECARBOXY AMIDE AND AN ARYL OR HETEROCYCLYL HALIDE OR A GROUP ENHANCING THE ELECTROPHILICITY OF THE ATOM TO WHICH IT IS ATTACHED FOR DISPLACEMENT; USING A PALLADIUM COMPOUND CATALYST, A BASE AND AN ACID ELI LILLY AND COMPANY (US) 2000-05-30 US disclosed
EP-0944581-A1 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES ELI LILLY AND COMPANY (US) 1999-09-29 EP disclosed
US-5917038-A REACTING PROPIOLAMIDE WITH ACTIVATED AROMATIC RING IN THE PRESENCE OF A PALLADIUM CATALYST ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed
WO-1998022429-A1 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES ELI LILLY AND COMPANY (US) 1998-05-28 WO disclosed