SCHEMBL6563222

SCHEMBL6563222

C#CC(=O)N(C)c1ccccc1C

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.45
ALDH1A1 P00352 1/20 0.44
HSD17B1 P14061 13/20 0.43
HSD17B2 P37059 11/20 0.43
GPBAR1 Q8TDU6 1/20 0.42
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12550525 0.79 ALDH1A1 (0.53) SIGMAR1ALDH1A1HSD17B1HSD17B2LMNA
Benzene SCHEMBL28335658 0.78 TRPM8 (0.50) SIGMAR1ALDH1A1HSD17B1HSD17B2LMNA
SCHEMBL1029152 0.78 TRPM8 (0.50) SIGMAR1ALDH1A1HSD17B1HSD17B2LMNA
SCHEMBL5042970 0.78 TSPO (0.53) SIGMAR1ALDH1A1HSD17B1HSD17B2LMNA
SCHEMBL2090213 0.78 HSD17B1 (0.49) SIGMAR1ALDH1A1HSD17B1HSD17B2LMNA
SCHEMBL29674730 0.78 TSPO (0.53) SIGMAR1ALDH1A1HSD17B1HSD17B2LMNA
SCHEMBL6561817 0.77 SIGMAR1 (0.61) SIGMAR1
SCHEMBL5932324 0.76 SIGMAR1 (0.47) SIGMAR1ALDH1A1HSD17B1HSD17B2LMNA
SCHEMBL7815992 0.76 SIGMAR1 (0.47) SIGMAR1ALDH1A1HSD17B1HSD17B2LMNA
SCHEMBL10943951 0.76 SIGMAR1 (0.47) SIGMAR1ALDH1A1HSD17B1HSD17B2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944581-A4 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES LILLY CO ELI (US) 2004-09-08 EP disclosed
US-6069247-A REACTING AN ACETYLENECARBOXY AMIDE AND AN ARYL OR HETEROCYCLYL HALIDE OR A GROUP ENHANCING THE ELECTROPHILICITY OF THE ATOM TO WHICH IT IS ATTACHED FOR DISPLACEMENT; USING A PALLADIUM COMPOUND CATALYST, A BASE AND AN ACID ELI LILLY AND COMPANY (US) 2000-05-30 US disclosed
EP-0944581-A1 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES ELI LILLY AND COMPANY (US) 1999-09-29 EP disclosed
US-5917038-A REACTING PROPIOLAMIDE WITH ACTIVATED AROMATIC RING IN THE PRESENCE OF A PALLADIUM CATALYST ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed
WO-1998022429-A1 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES ELI LILLY AND COMPANY (US) 1998-05-28 WO disclosed