SCHEMBL6561817

SCHEMBL6561817

C#CC(=O)N(C)c1cccc2ccccc12

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 12/20 0.61
CNR2 P34972 1/20 0.39
GAA P10253 2/20 0.39
TSHR P16473 1/20 0.39
NR4A1 P22736 1/20 0.39
NR4A2 P43354 1/20 0.39
NR4A3 Q92570 1/20 0.39
PLK1 P53350 1/20 0.39
MCL1 Q07820 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29666490 0.80 SIGMAR1 (0.67) SIGMAR1CNR2GAANR4A1NR4A2
SCHEMBL3626830 0.80 SIGMAR1 (0.67) SIGMAR1GAATSHRNR4A1NR4A2
SCHEMBL1614544 0.80 SIGMAR1 (0.67) SIGMAR1CNR2GAANR4A1NR4A2
SCHEMBL6560707 0.80 ALDH1A1 (0.39) SIGMAR1GAA
SCHEMBL10943508 0.79 SIGMAR1 (0.65) SIGMAR1CNR2GAANR4A1NR4A2
SCHEMBL1839015 0.79 SIGMAR1 (0.65) SIGMAR1GAA
SCHEMBL8150820 0.79 SIGMAR1 (0.65) SIGMAR1GAANR4A1NR4A2NR4A3
SCHEMBL11872011 0.79 SIGMAR1 (0.65) SIGMAR1CNR2GAANR4A1NR4A2
SCHEMBL28259034 0.79 SIGMAR1 (0.65) SIGMAR1CNR2GAANR4A1NR4A2
SCHEMBL6563222 0.77 SIGMAR1 (0.45) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944581-A4 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES LILLY CO ELI (US) 2004-09-08 EP disclosed
US-6069247-A REACTING AN ACETYLENECARBOXY AMIDE AND AN ARYL OR HETEROCYCLYL HALIDE OR A GROUP ENHANCING THE ELECTROPHILICITY OF THE ATOM TO WHICH IT IS ATTACHED FOR DISPLACEMENT; USING A PALLADIUM COMPOUND CATALYST, A BASE AND AN ACID ELI LILLY AND COMPANY (US) 2000-05-30 US disclosed
EP-0944581-A1 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES ELI LILLY AND COMPANY (US) 1999-09-29 EP disclosed
US-5917038-A REACTING PROPIOLAMIDE WITH ACTIVATED AROMATIC RING IN THE PRESENCE OF A PALLADIUM CATALYST ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed
WO-1998022429-A1 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES ELI LILLY AND COMPANY (US) 1998-05-28 WO disclosed