SCHEMBL6560871

SCHEMBL6560871

CC(C)C[C@H](N)C(=O)N[C@@H](CO)[C@@H](O)[C@@H](O)[C@H](O)C(=O)N[C@@H](CC(=O)N[C@@H](C)C(=O)O)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 3/20 0.45
METAP1 P53582 3/20 0.45
SCN9A Q15858 1/20 0.42
REN P00797 5/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
GPR88 Q9GZN0 2/20 0.37
MME P08473 2/20 0.36
LARS1 Q9P2J5 1/20 0.36
LTA4H P09960 1/20 0.36
ANPEP P15144 1/20 0.36
CTSD P07339 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6558600 0.92 METAP2 (0.44) METAP2METAP1SCN9AALDH1A1LMNA
SCHEMBL6559733 0.89 METAP2 (0.48) METAP2METAP1SCN9AALDH1A1LMNA
SCHEMBL6560489 0.88 METAP2 (0.47) METAP2METAP1SCN9AALDH1A1LMNA
Hydrochloric Acid SCHEMBL6559799 0.88 METAP2 (0.47) METAP2METAP1SCN9AALDH1A1LMNA
Hydrochloric Acid SCHEMBL6560650 0.86 METAP2 (0.45) METAP2METAP1SCN9ARENALDH1A1
SCHEMBL6559036 0.82 METAP2 (0.40) METAP2METAP1SCN9AALDH1A1LMNA
SCHEMBL6559229 0.81 METAP2 (0.45) METAP2METAP1SCN9AMMECTSD
SCHEMBL6558906 0.81 PSMB1 (0.43) METAP2METAP1SCN9ACTSD
Hydrochloric Acid SCHEMBL6560661 0.81 KEAP1 (0.45) METAP2METAP1SCN9AMMELARS1
SCHEMBL6560842 0.80 METAP2 (0.43) METAP2METAP1SCN9AMMECTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998488-B1 POLYOL-AMINO ACID COMPOUNDS HAVING ANTI-HELICOBACTER PYLORI ACTIVITY TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2004-03-17 EP disclosed
US-6423869-B1 BACTERICIDES, ANTIULCER AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-07-23 US disclosed