SCHEMBL6563210

SCHEMBL6563210

COC(=O)[C@H](Cc1ccc(NC(=O)c2ccc(Cl)nc2Cl)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.46
TDP1 Q9NUW8 4/20 0.46
KDM4E B2RXH2 3/20 0.46
ITGB1 P05556 2/20 0.45
ITGB3 P05106 2/20 0.45
ITGA2B P08514 2/20 0.45
ITGAV P06756 1/20 0.45
ITGB5 P18084 1/20 0.45
KLK5 Q9Y337 1/20 0.45
NPSR1 Q6W5P4 4/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
HDAC8 Q9BY41 1/20 0.42
CTSS P25774 6/20 0.41
CTSK P43235 5/20 0.41
KLKB1 P03952 1/20 0.40
KLK1 P06870 1/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
XBP1 P17861 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6560946 0.87 MAPT (0.49) MAPTTDP1KDM4EITGB1ITGB3
SCHEMBL6561292 0.81 ITGB1 (0.56) ITGB1ITGB3ITGA2BITGAVITGB5
SCHEMBL14799578 0.81 ITGB1 (0.56) ITGB1ITGB3ITGA2BITGAVITGB5
SCHEMBL6642502 0.81 GAA (0.48) MAPTITGB1ITGB3ITGA2BITGAV
SCHEMBL27278646 0.80 KLK5 (0.54) MAPTTDP1KDM4EITGB1ITGB3
Hydrochloric Acid SCHEMBL6560412 0.79 PTGS2 (0.41) ITGB1KLKB1KLK1ITGA4
SCHEMBL20715930 0.79 ITGB3 (0.61) MAPTTDP1KDM4EITGB1ITGB3
SCHEMBL15140552 0.79 ITGB1 (0.48) MAPTTDP1KDM4EITGB1ITGB3
SCHEMBL15140555 0.79 ITGB1 (0.48) MAPTTDP1KDM4EITGB1ITGB3
SCHEMBL20865337 0.79 KLK5 (0.53) MAPTTDP1KDM4EITGB1ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144365-B1 INHIBITORS OF ALPHA-4 BETA-1 MEDIATED CELL ADHESION TANABE SEIYAKU CO (JP) 2004-03-17 EP disclosed