SCHEMBL6563346

SCHEMBL6563346

CNC(=O)/C=C(\c1ccc(C(F)(F)F)cc1)c1cccc(F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.45
MTOR P42345 1/20 0.45
HPGDS O60760 1/20 0.45
TRPV1 Q8NER1 1/20 0.43
KDR P35968 2/20 0.42
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 1/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
CES2 O00748 3/20 0.41
CES1 P23141 2/20 0.41
NR4A1 P22736 1/20 0.40
NR4A2 P43354 1/20 0.40
NR4A3 Q92570 1/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6561899 0.82 ALDH1A1 (0.60) KDM4EALDH1A1NPC1RAB9ALMNA
SCHEMBL6561870 0.82 ALDH1A1 (0.60) KDM4EALDH1A1NPC1RAB9ALMNA
SCHEMBL6563253 0.75 TSHR (0.45) KDM4ENPC1RAB9ACES2CES1
SCHEMBL6563249 0.75 TSHR (0.45) KDM4ENPC1RAB9ACES2CES1
SCHEMBL6561874 0.75 PLK1 (0.47) TRPV1ALDH1A1NPC1RAB9ANR4A1
SCHEMBL6562127 0.75 PLK1 (0.47) TRPV1ALDH1A1NPC1RAB9ANR4A1
SCHEMBL3945565 0.74 MAOB (0.43) MAOBMTORHPGDSALDH1A1CES2
SCHEMBL3945568 0.74 MAOB (0.43) MAOBMTORHPGDSALDH1A1CES2
SCHEMBL3945561 0.74 MAOB (0.43) MAOBMTORHPGDSALDH1A1CES2
SCHEMBL6561880 0.73 PLK1 (0.48) KDM4ENPC1RAB9ACES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944581-A4 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES LILLY CO ELI (US) 2004-09-08 EP disclosed
EP-0944581-A1 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES ELI LILLY AND COMPANY (US) 1999-09-29 EP disclosed
WO-1998022429-A1 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES ELI LILLY AND COMPANY (US) 1998-05-28 WO disclosed