SCHEMBL6563559

SCHEMBL6563559

CCOC(=O)CN(C(=O)Nc1cc(C(F)(F)F)c(C#CCNc2ccc(C(=N)N)cc2)cc1C)C(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.36
ITGA2B P08514 2/20 0.36
F7 P08709 4/20 0.34
F2 P00734 11/20 0.32
IDH1 O75874 2/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.31
RAB9A P51151 1/20 0.31
PAX8 Q06710 1/20 0.31
F10 P00742 8/20 0.31
PRSS1 P07477 5/20 0.30
KLK1 P06870 1/20 0.30
PLAU P00749 1/20 0.30
PLAT P00750 1/20 0.30
PRSS2 P07478 1/20 0.30
F3 P13726 1/20 0.30
PRSS3 P35030 1/20 0.30
NQO2 P16083 1/20 0.30
PLG P00747 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6565445 0.95 ITGB3 (0.36) ITGB3ITGA2BF7F2NPC1
SCHEMBL6563746 0.91 F7 (0.37) ITGB3ITGA2BF7F2NPC1
SCHEMBL7670894 0.91 ITGB3 (0.39) ITGB3ITGA2BF7F2F10
SCHEMBL6565368 0.90 ITGB3 (0.37) ITGB3ITGA2BF7F2IDH1
SCHEMBL6563523 0.88 ITGB3 (0.37) ITGB3ITGA2BF7F2RAB9A
SCHEMBL6565399 0.85 ITGB3 (0.37) ITGB3ITGA2BF7F2F10
SCHEMBL6563598 0.84 F7 (0.38) ITGB3ITGA2BF7F2NPC1
SCHEMBL6563366 0.84 ITGB3 (0.39) ITGB3ITGA2BF7F2ALDH1A1
SCHEMBL6563089 0.84 PLAU (0.33) ITGB3ITGA2BF7F2F10
SCHEMBL6561894 0.84 ITGB3 (0.40) ITGB3ITGA2BF7F2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed